SCHEMBL907644

SCHEMBL907644

COc1nc(C)ncc1OC(C)=O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TNFSF11 O14788 1/20 0.40
ALDH1A1 P00352 1/20 0.39
F2 P00734 1/20 0.39
GLA P06280 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 2/20 0.36
BACE1 P56817 1/20 0.36
KMT2A Q03164 1/20 0.36
PTPN1 P18031 1/20 0.36
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
POLB P06746 2/20 0.33
NR3C1 P04150 1/20 0.33
NQO1 P15559 1/20 0.33
KDM4E B2RXH2 1/20 0.33
JUN P05412 1/20 0.33
NFKB1 P19838 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16742632 0.80 HTT (0.38) TNFSF11ALDH1A1F2GLAHPGD
SCHEMBL10304905 0.79 KMT2A (0.52) ALDH1A1KMT2ASMN1; SMN2KDM4E
SCHEMBL5494945 0.79 HTT (0.37) TNFSF11ALDH1A1F2GLAHPGD
SCHEMBL5501359 0.77 KDM4E (0.41) ALDH1A1GLAHPGDTSHRKMT2A
SCHEMBL4046039 0.77 LMNA (0.42) TNFSF11ALDH1A1F2GLAHPGD
SCHEMBL907751 0.74 TNFSF11 (0.41) TNFSF11ALDH1A1F2GLAHPGD
SCHEMBL20116948 0.73 KMT2A (0.39) ALDH1A1HPGDTSHRKMT2ASMN1; SMN2
SCHEMBL20855865 0.71 HCRTR1 (0.42) ALDH1A1GLAHPGDTSHRKMT2A
SCHEMBL20524652 0.71 TDP1 (0.51) ALDH1A1HPGDKMT2AHTTSMN1; SMN2
SCHEMBL9814546 0.70 TNFSF11 (0.53) TNFSF11ALDH1A1F2GLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2276756-B1 HYDROXYMETHYL PYRROLIDINES AS BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME (US) 2011-11-30 EP disclosed
EP-2276756-A1 HYDROXYMETHYL PYRROLIDINES AS BETA 3 ADRENERGIC RECEPTOR AGONISTS Merck Sharp & Dohme Corp. (US) 2011-01-26 EP disclosed
EP-2274296-A1 HYDROXYMETHYL PYRROLIDINES AS BETA 3 ADRENERGIC RECEPTOR AGONISTS Merck Sharp & Dohme Corp. (US) 2011-01-19 EP disclosed