SCHEMBL9078917

SCHEMBL9078917

COC(=O)C(Cc1ccc(CC(=O)O)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.58
CTSS P25774 7/20 0.54
CTSK P43235 6/20 0.54
CTSB P07858 2/20 0.53
CTSL P07711 1/20 0.53
ACE P12821 1/20 0.51
ITGB3 P05106 1/20 0.51
ITGA2B P08514 1/20 0.51
ATM Q13315 1/20 0.47
EPHX2 P34913 1/20 0.47
ITGA4 P13612 1/20 0.47
ITGB7 P26010 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
AKT1 P31749 1/20 0.47
PPARA Q07869 2/20 0.46
PPARG P37231 1/20 0.46
MDM4 O15151 1/20 0.46
MDM2 Q00987 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9078913 1.00 KLK5 (0.58) KLK5CTSSCTSKCTSBCTSL
SCHEMBL9076747 0.90 KLK5 (0.56) KLK5CTSSCTSKCTSBCTSL
SCHEMBL9076749 0.90 KLK5 (0.56) KLK5CTSSCTSKCTSBCTSL
SCHEMBL7544681 0.88 KLK5 (0.57) KLK5CTSSCTSKCTSBCTSL
SCHEMBL6292728 0.88 KLK5 (0.72) KLK5CTSSCTSKCTSBCTSL
SCHEMBL84524 0.88 KLK5 (0.72) KLK5CTSSCTSKCTSBCTSL
SCHEMBL1196457 0.88 KLK5 (0.72) KLK5CTSSCTSKCTSBCTSL
SCHEMBL21473748 0.88 KLK5 (0.72) KLK5CTSSCTSKCTSBCTSL
SCHEMBL1826757 0.87 CTSS (0.69) KLK5CTSSCTSKCTSBCTSL
SCHEMBL10033679 0.87 CTSS (0.69) KLK5CTSSCTSKCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5508437-A APPETITE SUPPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-04-16 US claimed
US-5508437-A APPETITE SUPPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-04-16 US disclosed
US-5296608-A Intermediates for analogs of tyrosine sulfate or tyrosine phosphate containing peptides HOFFMAN-LA ROCHE INC. (US) 1994-03-22 US disclosed
US-5182263-A Appetite suppressants HOFFMANN-LA ROCHE INC. (US) 1993-01-26 US disclosed
EP-0339549-A2 Tyr-peptide analogs F. HOFFMANN-LA ROCHE AG (CH) 1989-11-02 EP disclosed