SCHEMBL9079018

SCHEMBL9079018

COc1cc2cc3c4c(cccc4c2cc1OC)C(=O)OC3=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.49
MEN1 O00255 4/20 0.49
POLB P06746 2/20 0.49
TYMS P04818 4/20 0.44
PRMT1 Q99873 1/20 0.42
KDM4E B2RXH2 4/20 0.41
MAPT P10636 4/20 0.41
ALDH1A1 P00352 3/20 0.41
LMNA P02545 2/20 0.41
PABPC1 P11940 1/20 0.41
XBP1 P17861 1/20 0.41
NFKB1 P19838 1/20 0.41
HTT P42858 1/20 0.41
SMARCA2 P51531 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
AHR P35869 1/20 0.41
NPC1 O15118 1/20 0.40
MAOA P21397 1/20 0.40
PDE1A P54750 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9080103 0.81 ALOX5 (0.44) KMT2AMEN1POLBTYMSKDM4E
SCHEMBL7709465 0.79 POLB (0.51) KMT2AMEN1POLBTYMSPRMT1
SCHEMBL30761754 0.78 KMT2A (0.76) KMT2AMEN1POLBTYMSPRMT1
SCHEMBL6548245 0.78 KMT2A (0.76) KMT2AMEN1POLBTYMSPRMT1
SCHEMBL9041820 0.76 ALDH1A1 (0.63) TYMSALDH1A1AHRMAOAHSD17B10
SCHEMBL9080061 0.76 TYMS (0.46) TYMSALDH1A1MAOAHSD17B10HPGD
SCHEMBL5256291 0.75 MCL1 (0.46) KMT2AMEN1POLBKDM4EMAPT
SCHEMBL7706740 0.74 KMT2A (0.47) KMT2AMEN1POLBTYMSPRMT1
SCHEMBL7712218 0.73 KMT2A (0.46) KMT2AMEN1POLBTYMSPRMT1
SCHEMBL9078978 0.73 TYMS (0.46) TYMSKDM4EALDH1A1HTTAHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585382-A ANTICARCINOGENIC AGENTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-17 US disclosed
CN-1125943-A Diimide polycyclic and heterocyclic chromophores as antitumor agents DU PONT MERCK PHARMA (US) 1996-07-03 CN disclosed
US-5416089-A Antitumor agent THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-05-16 US disclosed
WO-1995000490-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-01-05 WO disclosed