SCHEMBL9082178

SCHEMBL9082178

CC1(C)CN=C(c2ccc(N)c(O)c2)NC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
ALOX15 P16050 1/20 0.46
HSD17B10 Q99714 1/20 0.46
BRD4 O60885 1/20 0.38
MAP4K1 Q92918 3/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
PIK3CD O00329 2/20 0.32
ABL1 P00519 2/20 0.32
EGFR P00533 2/20 0.32
HCK P08631 2/20 0.32
SRC P12931 2/20 0.32
KDR P35968 2/20 0.32
PIK3CA P42336 2/20 0.32
PIK3CB P42338 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9083000 0.90 ALDH1A1 (0.39) CYP3A4ALOX15HSD17B10MAP4K1KDM4E
SCHEMBL9023407 0.86 TDP1 (0.41) CYP3A4ALOX15HSD17B10MAP4K1KDM4E
SCHEMBL14029047 0.81 NISCH (0.41) NISCH
SCHEMBL9023749 0.77 MAPT (0.53) CYP3A4ALOX15MEN1POLBGAA
SCHEMBL9082242 0.76 ALDH1A1 (0.43) ALOX15HSD17B10KDM4EMEN1POLB
SCHEMBL9082170 0.75 NISCH (0.53) CYP3A4ALOX15HSD17B10NISCH
SCHEMBL14854498 0.70 PRMT1 (0.45) KDM4EMAPTRAB9A
SCHEMBL24312945 0.70 ALOX5 (0.47) HSD17B10KDM4EMEN1GAAMAPT
SCHEMBL9112216 0.68 NPC1 (0.33) POLBGAAMAPTRAB9AEGFR
SCHEMBL2237656 0.68 ADRB2 (0.41) CYP3A4KDM4EGAAMAPTNISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996028443-A1 THERAPEUTIC BENZOXAZOLES THE WELLCOME FOUNDATION LIMITED (GB) 1996-09-19 WO disclosed