SCHEMBL908524

SCHEMBL908524

OCCc1ccc(Cl)c(Cl)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.61
TAAR1 Q96RJ0 1/20 0.61
IGF1R P08069 1/20 0.57
ALOX15 P16050 1/20 0.57
IDO1 P14902 3/20 0.54
SIGMAR1 Q99720 11/20 0.53
ALDH1A1 P00352 2/20 0.52
MAPT P10636 2/20 0.52
KDM4E B2RXH2 1/20 0.52
ALOX5 P09917 1/20 0.52
GAA P10253 1/20 0.52
BACE1 P56817 1/20 0.52
CYP1A2 P05177 2/20 0.48
MEN1 O00255 1/20 0.48
TP53 P04637 1/20 0.48
CYP2C19 P33261 1/20 0.48
KMT2A Q03164 1/20 0.48
PYGL P06737 1/20 0.47
CYP2D6 P10635 1/20 0.47
TMEM97 Q5BJF2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL81497 0.86 IGF1R (0.63) PNMTTAAR1IGF1RALOX15IDO1
SCHEMBL9026682 0.85 IGF1R (0.67) PNMTTAAR1IGF1RALOX15IDO1
SCHEMBL10609252 0.83 IGF1R (0.65) PNMTTAAR1IGF1RALOX15IDO1
SCHEMBL8905783 0.83 IGF1R (0.65) PNMTTAAR1IGF1RALOX15IDO1
SCHEMBL7008253 0.83 IGF1R (0.65) PNMTTAAR1IGF1RALOX15IDO1
SCHEMBL25218464 0.82 ALDH1A1 (0.65) PNMTTAAR1IGF1RALOX15ALDH1A1
SCHEMBL5454185 0.82 KDM4E (0.65) IGF1RALOX15ALDH1A1MAPTKDM4E
SCHEMBL2299809 0.80 ALDH1A1 (0.47) PNMTTAAR1IGF1RALOX15IDO1
SCHEMBL12333663 0.80 ALDH1A1 (0.47) PNMTTAAR1IGF1RALOX15ALDH1A1
SCHEMBL3264645 0.80 MAPT (0.47) PNMTTAAR1IGF1RALOX15ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 155 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0767174-A1 Novel aminoalkanephosphinic acids and their salts CIBA-GEIGY AG (CH) 1997-04-09 EP claimed
US-5376684-A Aminobutyric acid antagonist; antiepileptic agent CIBA-GEIGY CORPORATION (US) 1994-12-27 US claimed
EP-0543780-A2 Novel aminoalkanephosphinic acids and their salts CIBA-GEIGY AG (CH) 1993-05-26 EP claimed
US-12528773-B2 Non-lysosomal glucosylceramidase inhibitors and uses thereof ALECTOS THERAPEUTICS INC. (CA) 2026-01-20 US disclosed
CN-119546605-A Protein degradation agent 苏州开拓药业股份有限公司 2025-02-28 CN disclosed
WO-2024027694-A9 PROTEIN DEGRADATION AGENT 苏州开拓药业股份有限公司 2025-01-02 WO disclosed
US-20240228502-A1 2-PHENYLAMINO PYRROLOPYRIMIDINES AS ACK1 INHIBITORS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2024-07-11 US disclosed
WO-2024027795-A1 ANTIBODY-DRUG CONJUGATE CONTAINING MYC PROTEIN DEGRADATION AGENT BIOACTIVE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF 苏州开拓药业股份有限公司 2024-02-08 WO disclosed
WO-2024027694-A1 PROTEIN DEGRADATION AGENT 苏州开拓药业股份有限公司 2024-02-08 WO disclosed
US-11827637-B2 Azaindole derivatives and their use as ERK kinase inhibitors AGV DISCOVERY (FR) 2023-11-28 US disclosed
US-20230348387-A1 NON-LYSOSOMAL GLUCOSYLCERAMIDASE INHIBITORS AND USES THEREOF ALECTOS THERAPEUTICS INC. (CA) 2023-11-02 US disclosed
WO-1991019707-A2 ANTIATHEROSCLEROTIC AND ANTITHROMBOTIC 1-BENZOPYRAN-4-ONES AND 2-AMINO-1,3-BENZOXAZINE-4-ONES THE UPJOHN COMPANY (US) 1991-12-26 WO disclosed
EP-0459983-A1 ANTIATHEROSCLEROTIC AND ANTITHROMBOTIC 1-BENZOPYRAN-4-ONES AND 2-AMINO-1,3-BENZOXAZINE-4-ONES PHARMACIA & UPJOHN COMPANY (US) 1991-12-11 EP disclosed
EP-0256888-B1 BENZOTHIAZEPINE VASODILATORS HAVING ARALKYL SUBSTITUTION McNeilab, Inc. (US) 1991-07-03 EP disclosed
WO-1991009013-A1 MUSCARINIC RECEPTOR ANTAGONISTS PFIZER LIMITED (GB) 1991-06-27 WO disclosed
EP-0411150-A1 INDOLE DERIVATIVES, PREPARATION THEREOF, AND DRUG FOR PREVENTING AND TREATING NEPHRITIS CONTAINING SAME OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-02-06 EP disclosed
WO-1990006921-A1 ANTIATHEROSCLEROTIC AND ANTITHROMBOTIC 1-BENZOPYRAN-4-ONES AND 2-AMINO-1,3-BENZOXAZINE-4-ONES THE UPJOHN COMPANY (US) 1990-06-28 WO disclosed
EP-0162208-B1 NOVEL N-SUBSTITUTED 3,4-DIHYDROPYRIMIDINE DERIVATIVES, PROCESSES FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS SUNTORY KABUSHIKI KAISHA, also known as SUNTORY LTD. (JP) 1989-11-23 EP disclosed
US-4729994-A Benzothiazepine vasodilators having aralkyl substitution MCNEILAB, INC. (US) 1988-03-08 US disclosed
EP-0256888-A1 Benzothiazepine vasodilators having aralkyl substitution McNeilab, Inc. (US) 1988-02-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230348387-A1 NON-LYSOSOMAL GLUCOSYLCERAMIDASE INHIBITORS AND USES THEREOF GBA1, GBA2, GAA PNMT 3313/4885TAAR1 4166/4885IGF1R 2487/4885
US-20240228502-A1 2-PHENYLAMINO PYRROLOPYRIMIDINES AS ACK1 INHIBITORS ADCK1, DCK, TNKS2 PNMT 4186/4885TAAR1 4717/4885IGF1R 2212/4885
US-12528773-B2 Non-lysosomal glucosylceramidase inhibitors and uses thereof GBA1, GBA2, GAA PNMT 4179/4885TAAR1 3606/4885IGF1R 1099/4885
US-11827637-B2 Azaindole derivatives and their use as ERK kinase inhibitors MAPKAPK2, MAPK1, MAPK7 PNMT 721/4885TAAR1 1183/4885IGF1R 1133/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.