SCHEMBL9099992

SCHEMBL9099992

C1=COc2ncccc2N1

nearest known ligand 0.31

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
CYP1A2 P05177 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30931514 1.00 CA12 (0.31) CA12CA1CA2CA9CYP1A2
SCHEMBL2035350 1.00 CA12 (0.31) CA12CA1CA2CA9CYP1A2
SCHEMBL2518471 0.74 TDP2 (0.37) CA12CA1CA2CA9CYP1A2
SCHEMBL30047476 0.68
SCHEMBL1762427 0.68 NPC1 (0.35) CYP1A2SMN1; SMN2
SCHEMBL5530115 0.67 NPC1 (0.40) CYP1A2SMN1; SMN2
SCHEMBL924457 0.67 OTUD7B (0.31) CA12CA1CA2CA9
SCHEMBL16430005 0.67 CA12 (0.30) CA12CA1CA2CA9
SCHEMBL924702 0.67 CA12 (0.30) CA12CA1CA2CA9
SCHEMBL224635 0.66 ALOX5 (0.41) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0701560-A1 BICYCLIC ETHER DERIVATIVES AND THEIR USE AS 5-LIPOXYGENASE INHIBITORS ZENECA LIMITED (GB) 1996-03-20 EP disclosed
WO-1995030668-A1 CYCLIC ETHER DERIVATIVES AND PHARMACEUTICAL COMPOSITION CONTAINING THEM ZENECA LIMITED (GB) 1995-11-16 WO disclosed
WO-1994027999-A1 BICYCLIC ETHER DERIVATIVES AND THEIR USE AS 5-LIPOXYGENASE INHIBITORS ZENECA LIMITED (GB) 1994-12-08 WO disclosed
WO-1994025453-A1 4-ARYL-4-HYDROXY-TETRAHYDROPYRANS AND 3-ARYL-3-HYDROXY-TETRAHYDROFURANS AS 5-LIPOXYGENASE INHIBITORS ZENECA LIMITED (GB) 1994-11-10 WO disclosed