SCHEMBL9105568

SCHEMBL9105568

CCC(C=O)N(CCc1ccc(Cl)cc1)C(=O)CC1C(=O)N(C(Cl)Cc2ccc(Cl)cc2)CC(=O)N1CCCN1CCOCC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 2/20 0.34
ALDH1A1 P00352 3/20 0.33
USP2 O75604 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
TSHR P16473 1/20 0.33
TP53 P04637 1/20 0.33
TBXA2R P21731 1/20 0.33
TBXAS1 P24557 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
PPARG P37231 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
C5AR1 P21730 1/20 0.32
TACR2 P21452 2/20 0.32
HRH3 Q9Y5N1 1/20 0.32
MMP2 P08253 1/20 0.32
MMP3 P08254 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
MRGPRX1 Q96LB2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9104196 0.89 MDM2 (0.35) MDM2ALDH1A1USP2NPSR1TSHR
SCHEMBL9105301 0.89 TACR2 (0.42) TACR2HRH3MMP2MMP9
SCHEMBL9104517 0.88 ALDH1A1 (0.35) MDM2ALDH1A1USP2NPSR1TSHR
SCHEMBL9107408 0.86 LMNA (0.32) ALDH1A1TP53LMNAKDM4E
SCHEMBL3705051 0.84 APAF1 (0.36) MDM2ALDH1A1USP2NPSR1TSHR
SCHEMBL3710700 0.83 MDM2 (0.38) MDM2ALDH1A1USP2TSHRTP53
SCHEMBL3701509 0.82 KDM4E (0.40) MDM2ALDH1A1PPARGNCOR2TACR2
SCHEMBL3695334 0.82 MDM2 (0.35) MDM2ALDH1A1USP2NPSR1TSHR
SCHEMBL3697424 0.82 APAF1 (0.34) MDM2ALDH1A1USP2NPSR1TSHR
SCHEMBL9101546 0.81 C5AR1 (0.39) ALDH1A1C5AR1TACR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2460798-A2 APAF-1 INHIBITOR COMPOUNDS Laboratorios SALVAT, S.A. (ES) 2012-06-06 EP disclosed