SCHEMBL9107930

SCHEMBL9107930

CC(C)(CC(=O)N[C@@H]1CSc2ccccc2N(Cc2ccc(-c3ccccc3NC(=O)NCCO)cc2)C1=O)NCc1ccco1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 4/20 0.44
XIAP P98170 1/20 0.40
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
AGTR1 P30556 1/20 0.38
F7 P08709 4/20 0.36
F3 P13726 4/20 0.36
F2 P00734 1/20 0.36
MAPT P10636 2/20 0.36
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
MME P08473 1/20 0.35
ACE P12821 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9108493 0.93 XIAP (0.42) GHSRXIAPTSHRMAPK1AGTR1
SCHEMBL9104616 0.91 GHSR (0.43) GHSRXIAPAGTR1F7F3
SCHEMBL9102903 0.91 GHSR (0.55) GHSRXIAPAGTR1F7F3
SCHEMBL9106865 0.90 XIAP (0.39) GHSRXIAPTSHRMAPK1AGTR1
SCHEMBL9103074 0.90 GHSR (0.44) GHSRXIAPAGTR1F7F3
SCHEMBL9105520 0.89 GHSR (0.57) GHSRXIAPTSHRMAPK1AGTR1
SCHEMBL7785751 0.88 GHSR (0.45) GHSRXIAPAGTR1F7F3
SCHEMBL9108628 0.87 GHSR (0.37) GHSRXIAPTSHRMAPK1AGTR1
SCHEMBL7791984 0.87 GHSR (0.50) GHSRXIAPAGTR1F7F3
SCHEMBL9105564 0.86 GHSR (0.54) GHSRXIAPAGTR1F7F3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430144-A E.g, N-(1-((2'-((methoxycarbonyl)amino)(1,1'-biphenyl)-4-yl) methyl)-2,3,4,5-tetrahydro-2-oxo-1H-1-benzazepin-3-yl)-3 ((fur-2-yl)methyl)amino-3-methylbutanamide MERCK & CO., INC. (US) 1995-07-04 US disclosed