SCHEMBL9108628

SCHEMBL9108628

CC(C)(CC(=O)N[C@@H]1CSc2ccccc2N(Cc2ccc(-c3ccccc3NC(=O)N3CCOCC3)cc2)C1=O)NCc1ccco1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 4/20 0.37
AGTR1 P30556 1/20 0.37
XIAP P98170 1/20 0.37
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
F7 P08709 4/20 0.35
F3 P13726 4/20 0.35
F2 P00734 1/20 0.35
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TP53 P04637 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9108493 0.89 XIAP (0.42) GHSRAGTR1XIAPTSHRMAPK1
SCHEMBL9106865 0.89 XIAP (0.39) GHSRAGTR1XIAPTSHRMAPK1
SCHEMBL9104558 0.89 GHSR (0.48) GHSRAGTR1XIAPTSHRMAPK1
SCHEMBL7791696 0.89 XIAP (0.41) GHSRAGTR1XIAPF7F3
SCHEMBL7785876 0.88 GHSR (0.47) GHSRAGTR1XIAPTSHRF7
SCHEMBL9107930 0.87 GHSR (0.44) GHSRAGTR1XIAPTSHRMAPK1
SCHEMBL9105226 0.84 GHSR (0.42) GHSRAGTR1XIAPF7F3
SCHEMBL9105221 0.84 GHSR (0.42) GHSRAGTR1XIAPF7F3
SCHEMBL9107838 0.83 GHSR (0.41) GHSRAGTR1XIAPTSHRMAPK1
SCHEMBL9106413 0.83 GHSR (0.41) GHSRAGTR1XIAPF7F3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430144-A E.g, N-(1-((2'-((methoxycarbonyl)amino)(1,1'-biphenyl)-4-yl) methyl)-2,3,4,5-tetrahydro-2-oxo-1H-1-benzazepin-3-yl)-3 ((fur-2-yl)methyl)amino-3-methylbutanamide MERCK & CO., INC. (US) 1995-07-04 US disclosed
WO-1995003290-A1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO., INC. (US) 1995-02-02 WO disclosed