SCHEMBL9117246

SCHEMBL9117246

CCC(C)(C)c1ccc(Oc2ccc(C(F)(F)F)cc2NC(=O)Nc2ccc(Oc3ccccc3)cc2)c(S(=O)(=O)O)c1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 11/20 0.52
IDH2 P48735 1/20 0.49
BRAF P15056 2/20 0.47
PTGES O14684 1/20 0.47
ALOX5 P09917 1/20 0.47
P2RY1 P47900 1/20 0.44
CYP2C9 P11712 1/20 0.43
IDO1 P14902 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9118064 0.94 PTGES (0.50) RAF1IDH2BRAFPTGESALOX5
SCHEMBL9118546 0.91 RAF1 (0.52) RAF1BRAFPTGESALOX5P2RY1
SCHEMBL8432579 0.88 PTGES (0.58) IDH2PTGESALOX5
SCHEMBL8433479 0.87 PTGES (0.49) RAF1IDH2BRAFPTGESALOX5
SCHEMBL9117651 0.85 HTT (0.56) CYP2C9
SCHEMBL9116337 0.84 P2RY1 (0.45) P2RY1IDO1
SCHEMBL9117910 0.84 PTGES (0.46) IDH2PTGESALOX5P2RY1
SCHEMBL8432745 0.84 PTGES (0.48) BRAFPTGESALOX5
SCHEMBL9243116 0.82 IDH2 (0.46) RAF1IDH2BRAFP2RY1CYP2C9
SCHEMBL9289620 0.80 PTGES (0.49) RAF1IDH2PTGESALOX5CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995033458-A1 ANTI-INFLAMMATORY COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-12-14 WO claimed
WO-1995033458-A1 ANTI-INFLAMMATORY COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-12-14 WO disclosed