SCHEMBL9243116

SCHEMBL9243116

CCC(C)(C)c1ccc(Oc2ccc(C(F)(F)F)cc2NC(=O)Nc2ccccc2)c(S)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDH2 P48735 1/20 0.46
HTT P42858 4/20 0.46
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
MAPT P10636 3/20 0.46
RAB9A P51151 2/20 0.46
RAF1 P04049 5/20 0.46
GRIK1 P39086 2/20 0.45
BRAF P15056 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
LMNA P02545 1/20 0.44
ATM Q13315 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
IDO1 P14902 1/20 0.43
P2RY1 P47900 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9118064 0.87 PTGES (0.50) IDH2HTTKMT2AMEN1MAPT
SCHEMBL8740768 0.85 KDR (0.50) RAF1BRAF
SCHEMBL9117246 0.82 RAF1 (0.52) IDH2RAF1BRAFCYP2C9IDO1
SCHEMBL9118596 0.81 GRIK1 (0.49) IDH2HTTKMT2AMEN1MAPT
SCHEMBL8432579 0.81 PTGES (0.58) IDH2HTTKMT2AMEN1MAPT
SCHEMBL9116521 0.79 KMT2A (0.42) HTTKMT2AMEN1MAPTCYP1A2
Diphenylmethanol SCHEMBL9188471 0.79 GRIK1 (0.45) IDH2HTTKMT2AMEN1MAPT
SCHEMBL8433479 0.78 PTGES (0.49) IDH2HTTKMT2AMEN1MAPT
SCHEMBL9119780 0.78 L3MBTL1 (0.43) IDH2HTTKMT2AMEN1MAPT
SCHEMBL5719998 0.78 CA12 (0.47) IDH2HTTKMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995033458-A1 ANTI-INFLAMMATORY COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-12-14 WO disclosed