SCHEMBL9118380

SCHEMBL9118380

COC(=O)c1ccccc1Oc1ccc(C(F)(F)F)cc1NC(=O)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 2/20 0.47
RAF1 P04049 2/20 0.47
RXFP1 Q9HBX9 2/20 0.47
IDH2 P48735 1/20 0.46
MAPT P10636 5/20 0.46
LMNA P02545 3/20 0.46
KDM4E B2RXH2 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
HTT P42858 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
ATM Q13315 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HPGD P15428 1/20 0.46
KDR P35968 1/20 0.46
CCR1 P32246 1/20 0.46
CCR2 P41597 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
POLB P06746 1/20 0.45
CCR6 P51684 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9117124 0.89 GRIK1 (0.58) GRIK1RXFP1IDH2MAPTHTT
SCHEMBL9119633 0.85 RXFP1 (0.45) GRIK1RAF1RXFP1MAPTLMNA
SCHEMBL9119627 0.81 GRIK1 (0.52) GRIK1RXFP1IDH2MAPTCCR1
SCHEMBL9118124 0.81 GRIK1 (0.61) GRIK1RXFP1MAPTHTTMEN1
SCHEMBL9117381 0.81 PTGES (0.52) GRIK1RAF1IDH2MAPTLMNA
SCHEMBL16302025 0.79 SCN8A (0.53) MAPTTDP1
SCHEMBL9186824 0.78 MAPT (0.53) GRIK1RAF1MAPTLMNAKDM4E
SCHEMBL5595139 0.78 CCR1 (0.54) GRIK1MAPTLMNANPSR1ATM
SCHEMBL9118596 0.78 GRIK1 (0.49) GRIK1RAF1IDH2MAPTLMNA
SCHEMBL9119563 0.77 RXFP1 (0.49) RXFP1MAPTLMNAKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995033460-A1 ANTI-INFLAMMATORY COUMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-12-14 WO claimed
US-5447957-A Anti-inflammatory compounds SMITHKLINE BEECHAM CORP. (US) 1995-09-05 US claimed
WO-1995033460-A1 ANTI-INFLAMMATORY COUMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-12-14 WO disclosed
US-5447957-A Anti-inflammatory compounds SMITHKLINE BEECHAM CORP. (US) 1995-09-05 US disclosed