SCHEMBL9118596

SCHEMBL9118596

CCC(C)(C)c1ccc(Oc2ccc(C(F)(F)F)cc2NC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c(C(=O)O)c1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 8/20 0.49
RAF1 P04049 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
IDO1 P14902 5/20 0.42
IDH2 P48735 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
ATM Q13315 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diphenylmethanol SCHEMBL9188471 0.92 GRIK1 (0.45) GRIK1CYP1A2CYP2C9IDO1IDH2
SCHEMBL9182258 0.91 GRIK1 (0.48) GRIK1RAF1CYP1A2CYP2C9CYP2C19
SCHEMBL9119780 0.86 L3MBTL1 (0.43) GRIK1RAF1CYP1A2CYP2C9IDO1
SCHEMBL8433479 0.85 PTGES (0.49) RAF1CYP1A2CYP2C9CYP2C19IDH2
SCHEMBL5719998 0.85 CA12 (0.47) RAF1CYP1A2CYP2C9CYP2C19IDH2
SCHEMBL9117124 0.83 GRIK1 (0.58) GRIK1IDH2MEN1KMT2AMAPT
SCHEMBL8081653 0.82 CCR2 (0.58) MEN1KMT2A
SCHEMBL9243116 0.81 IDH2 (0.46) GRIK1RAF1CYP1A2CYP2C9CYP2C19
SCHEMBL9186824 0.79 MAPT (0.53) GRIK1RAF1LMNAMAPT
SCHEMBL9118064 0.79 PTGES (0.50) GRIK1RAF1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5447957-A Anti-inflammatory compounds SMITHKLINE BEECHAM CORP. (US) 1995-09-05 US claimed
WO-1995033460-A1 ANTI-INFLAMMATORY COUMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-12-14 WO disclosed
US-5447957-A Anti-inflammatory compounds SMITHKLINE BEECHAM CORP. (US) 1995-09-05 US disclosed