SCHEMBL9119044

SCHEMBL9119044

CS(=O)(=O)c1ccc(C2=CCC=C2CCc2ccc(C(F)(F)F)cc2)cn1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.38
PTGS2 P35354 3/20 0.35
DAO P14920 1/20 0.34
CTSK P43235 1/20 0.34
MAOB P27338 1/20 0.34
PPARD Q03181 2/20 0.34
RORC P51449 1/20 0.33
LOXL2 Q9Y4K0 2/20 0.33
STAT3 P40763 1/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
POLB P06746 1/20 0.33
HTR2A P28223 1/20 0.33
KCNH2 Q12809 1/20 0.33
GPR119 Q8TDV5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9116580 0.90 KIF11 (0.39) KIF11PTGS2CTSKPPARDRORC
SCHEMBL9117083 0.89 KIF11 (0.43) KIF11PTGS2MAOBALOX5APFEN1
SCHEMBL9117872 0.88 HTR2A (0.45) PTGS2CTSKRORCHTR2AKCNH2
SCHEMBL8974709 0.85 PTGS2 (0.42) KIF11PTGS2CTSKLOXL2ALOX5AP
SCHEMBL8975024 0.80 PTGS2 (0.38) KIF11PTGS2CTSKLOXL2ALOX5AP
SCHEMBL9116165 0.79 KIF11 (0.44) KIF11PTGS2MAOBPPARDALOX5AP
SCHEMBL9276607 0.76 HTR2A (0.45) PTGS2MAOBHTR2AKCNH2
SCHEMBL8974062 0.73 KIF11 (0.45) KIF11PTGS2ALOX5APFEN1
SCHEMBL9118890 0.72 PTGS2 (0.48) KIF11PTGS2CTSKALOX5APFEN1
SCHEMBL8974150 0.72 ALOX5AP (0.40) KIF11PTGS2LOXL2ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed