SCHEMBL9119279

SCHEMBL9119279

Ic1ccc2c(c1)COCC2

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PNMT P11086 6/20 0.46
ADRA2A P08913 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46
TDP2 O95551 2/20 0.34
PIK3CD O00329 1/20 0.34
PIR O00625 1/20 0.32
HTR6 P50406 1/20 0.32
PRMT5 O14744 1/20 0.30
WDR77 Q9BQA1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13617231 0.92 PNMT (0.41) PNMTADRA2AADRA2BADRA2CTDP2
SCHEMBL10238388 0.82 PNMT (0.42) PNMTADRA2AADRA2BADRA2CTDP2
SCHEMBL29989368 0.75 MAPT (0.40) PIK3CDHTR6PRMT5WDR77
SCHEMBL9122886 0.75 CA1 (0.39) PIK3CDHTR6
SCHEMBL31246225 0.75 CA1 (0.39) PIK3CDHTR6
SCHEMBL29790845 0.75 PNMT (0.46) PNMTADRA2AADRA2BADRA2CTDP2
SCHEMBL4523516 0.75 PNMT (0.46) PNMTADRA2AADRA2BADRA2CTDP2
SCHEMBL19023151 0.75 DRD2 (0.43)
SCHEMBL8237889 0.75 PIK3CD (0.36) ADRA2APIK3CDPIR
SCHEMBL9125380 0.75 HTR2A (0.48) PNMTADRA2AADRA2BADRA2CPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021048567-A1 NEW COMPOUNDS AND METHODS BENEVOLENTAI BIO LIMITED (GB) 2021-03-18 WO disclosed
US-5395827-A Analgesic, anticonvulsant, antiepileptic and anxiolytic agents GUILFORD PHARMACEUTICALS INC. (US) 1995-03-07 US disclosed
US-5364876-A Tranquilizers, analgesics, learning enhancement GUILFORD PHARMACEUTICALS INC. (US) 1994-11-15 US disclosed
WO-1993005772-A1 φ-[2-(PHOSPHONOALKYL)PHENYL]-2-AMINOALKANOIC ACIDS AS ANTAGONISTS OF EXCITATORY AMINO ACID RECEPTORS NOVA PHARMACEUTICAL CORPORATION (US) 1993-04-01 WO disclosed