SCHEMBL9124787

SCHEMBL9124787

COc1ccc(COc2cccnc2NC(=N)Nc2ccc(Cl)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PPIA P62937 12/20 0.60
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
GAA P10253 2/20 0.53
MAPT P10636 2/20 0.53
KDM4E B2RXH2 1/20 0.53
LMNA P02545 1/20 0.53
POLB P06746 1/20 0.53
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
FPR2 P25090 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PPIF P30405 1/20 0.44
ALDH1A1 P00352 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
KDR P35968 1/20 0.43
CNR1 P21554 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9122331 0.90 PPIA (0.61) PPIAMEN1KMT2AGAAMAPT
SCHEMBL9128497 0.90 PPIA (0.60) PPIAMEN1KMT2AMAPTNPC1
SCHEMBL9125073 0.89 PPIA (0.75) PPIAPPIF
SCHEMBL9125085 0.89 PPIA (0.68) PPIAPPIF
SCHEMBL9122377 0.87 PPIA (0.60) PPIAMEN1KMT2AGAAMAPT
SCHEMBL9126091 0.85 PPIA (0.46) PPIAMEN1KMT2AGAAMAPT
SCHEMBL9127894 0.81 PPIA (0.55) PPIAKMT2AMAPTLMNAPOLB
SCHEMBL9126123 0.80 PPIA (0.54) PPIAMEN1KMT2ANPC1RAB9A
SCHEMBL9124958 0.80 PPIA (0.56) PPIAGAAMAPTNPC1RAB9A
SCHEMBL2783281 0.80 PPIA (0.72) PPIAPPIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed