SCHEMBL9127894

SCHEMBL9127894

N=C(Nc1ccc(Cl)cc1)Nc1ncccc1OCc1c(Cl)cccc1Cl

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPIA P62937 10/20 0.55
SGMS2 Q8NHU3 3/20 0.45
SGMS1 Q86VZ5 1/20 0.43
PPIF P30405 2/20 0.41
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
AKR1C3 P42330 1/20 0.39
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9127827 0.92 PPIA (0.50) PPIASGMS2PPIFRAB9ASMN1; SMN2
SCHEMBL9126609 0.92 PPIA (0.53) PPIASGMS2SGMS1PPIF
SCHEMBL9124032 0.89 PPIA (0.53) PPIASGMS2PPIFRAB9ANPC1
SCHEMBL9124958 0.87 PPIA (0.56) PPIASGMS2SGMS1PPIFRAB9A
SCHEMBL9129017 0.87 SGMS2 (0.50) PPIASGMS2PPIFRAB9ASMN1; SMN2
SCHEMBL9124740 0.86 PPIA (0.55) PPIASGMS2SGMS1RAB9ANPC1
SCHEMBL9125346 0.86 PPIA (0.50) PPIASGMS2SGMS1PPIFRAB9A
SCHEMBL9128706 0.85 PPIA (0.52) PPIASGMS2PPIFRAB9ANPC1
SCHEMBL9125073 0.85 PPIA (0.75) PPIAPPIF
SCHEMBL9126729 0.84 SGMS2 (0.55) PPIASGMS2PPIFRAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed