SCHEMBL9124958

SCHEMBL9124958

N=C(Nc1ccc(Cl)cc1)Nc1ncccc1OCc1ccccc1Cl

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PPIA P62937 10/20 0.56
SGMS2 Q8NHU3 3/20 0.47
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
THRB P10828 1/20 0.46
SGMS1 Q86VZ5 1/20 0.43
PPIF P30405 2/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LRRK2 Q5S007 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9125346 0.89 PPIA (0.50) PPIASGMS2GAAMAPTTHRB
SCHEMBL9126123 0.89 PPIA (0.54) PPIASGMS2SGMS1NPC1RAB9A
SCHEMBL9127894 0.87 PPIA (0.55) PPIASGMS2MAPTSGMS1PPIF
SCHEMBL9126341 0.86 PPIA (0.56) PPIASGMS2GAAMAPTTHRB
SCHEMBL9125073 0.86 PPIA (0.75) PPIAPPIF
SCHEMBL9125085 0.84 PPIA (0.68) PPIAPPIF
SCHEMBL9127445 0.83 PPIA (0.48) PPIASGMS2PPIFNPC1RAB9A
SCHEMBL9124706 0.83 PPIA (0.50) PPIASGMS2PPIF
SCHEMBL9127827 0.83 PPIA (0.50) PPIASGMS2PPIFRAB9ASMN1; SMN2
SCHEMBL9126609 0.81 PPIA (0.53) PPIASGMS2SGMS1PPIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed