SCHEMBL9126123

SCHEMBL9126123

Cc1ccccc1COc1cccnc1NC(=N)Nc1ccc(Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPIA P62937 10/20 0.54
RAB9A P51151 2/20 0.48
SGMS2 Q8NHU3 4/20 0.45
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
NPC1 O15118 1/20 0.43
SGMS1 Q86VZ5 1/20 0.42
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
AKR1C3 P42330 1/20 0.41
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9123645 0.91 PPIA (0.52) PPIARAB9ASGMS2NPC1SGMS1
SCHEMBL9127445 0.90 PPIA (0.48) PPIARAB9ASGMS2MEN1CYP1A2
SCHEMBL9124958 0.89 PPIA (0.56) PPIARAB9ASGMS2NPC1SGMS1
SCHEMBL9126340 0.87 PPIA (0.54) PPIARAB9ASGMS2MEN1CYP1A2
SCHEMBL9125073 0.84 PPIA (0.75) PPIA
SCHEMBL9125096 0.84 PPIA (0.51) PPIARAB9ASGMS2MEN1CYP1A2
SCHEMBL9122331 0.83 PPIA (0.61) PPIARAB9AMEN1KMT2A
SCHEMBL9125346 0.83 PPIA (0.50) PPIARAB9ASGMS2NPC1SGMS1
SCHEMBL9125085 0.82 PPIA (0.68) PPIA
SCHEMBL9127894 0.81 PPIA (0.55) PPIARAB9ASGMS2CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP claimed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO claimed
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed