SCHEMBL9124706

SCHEMBL9124706

N=C(Nc1ccc(Cl)cc1)Nc1ncccc1OCc1ccc(F)cc1F

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PPIA P62937 8/20 0.50
PTGER1 P34995 9/20 0.45
PPIF P30405 1/20 0.45
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
SGMS2 Q8NHU3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9126091 0.89 PPIA (0.46) PPIAPPIFSGMS2
SCHEMBL9125540 0.88 PPIA (0.50) PPIAPTGER1PPIF
SCHEMBL9124032 0.84 PPIA (0.53) PPIAPPIFSGMS2
SCHEMBL9125346 0.83 PPIA (0.50) PPIAPPIFSGMS2
SCHEMBL9127827 0.83 PPIA (0.50) PPIAPPIFSGMS2
SCHEMBL9128706 0.83 PPIA (0.52) PPIAPPIFSGMS2
SCHEMBL9124958 0.83 PPIA (0.56) PPIAPPIFSGMS2
SCHEMBL9127445 0.82 PPIA (0.48) PPIAPPIFCYP2C19SGMS2
SCHEMBL9127894 0.81 PPIA (0.55) PPIAPPIFCYP2C9CYP2C19SGMS2
SCHEMBL9126123 0.81 PPIA (0.54) PPIACYP2C19SGMS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed