SCHEMBL9126643

SCHEMBL9126643

CN(C(=N)Nc1ncccc1OCc1c(F)cccc1F)c1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPIF P30405 1/20 0.44
PPIA P62937 8/20 0.42
SGMS2 Q8NHU3 2/20 0.38
GUCY1B2 O75343 3/20 0.34
GUCY1A2 P33402 3/20 0.34
GUCY1A1 Q02108 3/20 0.34
GUCY1B1 Q02153 3/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
ERBB2 P04626 1/20 0.33
EPHA2 P29317 1/20 0.33
KDR P35968 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9126603 0.88 SGMS2 (0.47) PPIFPPIASGMS2TDP1ALDH1A1
SCHEMBL9124032 0.81 PPIA (0.53) PPIFPPIASGMS2ERBB2EPHA2
SCHEMBL9125551 0.77 PPIA (0.53) PPIFPPIASGMS2ALDH1A1KMT2A
SCHEMBL9357599 0.76 PPIA (0.50) PPIFPPIASGMS2ERBB2EPHA2
SCHEMBL9127827 0.76 PPIA (0.50) PPIFPPIASGMS2TDP1ALDH1A1
SCHEMBL9357595 0.76 PPIF (0.46) PPIFPPIASGMS2GUCY1B2GUCY1A2
SCHEMBL9124036 0.75 PPIF (0.48) PPIFPPIASGMS2GUCY1B2GUCY1A2
SCHEMBL9128706 0.74 PPIA (0.52) PPIFPPIASGMS2ALDH1A1KMT2A
Hydrochloric Acid SCHEMBL9126773 0.73 PPIA (0.48) PPIFPPIA
SCHEMBL9124294 0.72 PPIA (0.50) PPIFPPIASGMS2TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed