SCHEMBL9128573

SCHEMBL9128573

O=C(O)C(Cl)C(=O)c1ccc(Cl)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 2/20 0.43
KCNQ2 O43526 2/20 0.43
KCNE1 P15382 2/20 0.43
KCNQ1 P51787 2/20 0.43
KCNQ5 Q9NR82 1/20 0.43
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
CES2 O00748 2/20 0.40
CES1 P23141 2/20 0.40
TSHR P16473 1/20 0.40
S1PR1 P21453 1/20 0.39
S1PR3 Q99500 1/20 0.39
KMO O15229 4/20 0.38
MAOB P27338 2/20 0.36
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36
CHRNB2 P17787 1/20 0.36
SLC6A2 P23975 1/20 0.36
CHRNB4 P30926 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9226597 0.86 CES2 (0.54) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL27243952 0.82 CES2 (0.49) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL8301590 0.81 KCNQ3 (0.42) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL8875867 0.81 KCNQ3 (0.43) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL28476035 0.81 KCNQ3 (0.44) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL29037468 0.80 KCNQ3 (0.42) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL4714984 0.79 KCNQ3 (0.38) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL479072 0.77 TSHR (0.65) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL27265284 0.77 S1PR1 (0.45) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL9860507 0.77 KCNQ3 (0.41) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5385906-A Treating gramnegative and grampositive bacterial infections THE UPJOHN COMPANY (US) 1995-01-31 US disclosed