SCHEMBL9128795

SCHEMBL9128795

CC(C)=CCCC(C)=Cc1ccc(C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.53
ALDH1A1 P00352 2/20 0.53
GLA P06280 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
RARB P10826 2/20 0.48
RARG P13631 2/20 0.48
RARA P10276 1/20 0.48
RXRA P19793 1/20 0.48
KDM4E B2RXH2 1/20 0.47
ATM Q13315 1/20 0.47
TRPV1 Q8NER1 3/20 0.47
ICMT O60725 1/20 0.44
GMNN O75496 1/20 0.44
TRPA1 O75762 1/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9128784 1.00 POLB (0.53) POLBALDH1A1GLATDP1L3MBTL1
SCHEMBL11052318 0.97 POLB (0.50) POLBALDH1A1GLATDP1L3MBTL1
SCHEMBL9288443 0.97 POLB (0.50) POLBALDH1A1GLATDP1L3MBTL1
SCHEMBL10486138 0.86 TRPV1 (0.46) POLBALDH1A1KDM4EATMTRPV1
SCHEMBL10485741 0.85 KDM4E (0.54) POLBALDH1A1KDM4EATMTRPV1
SCHEMBL11053782 0.84 LMNA (0.54) POLBALDH1A1GLATDP1L3MBTL1
SCHEMBL11053785 0.84 LMNA (0.54) POLBALDH1A1GLATDP1L3MBTL1
SCHEMBL9309827 0.82 UNG (0.49) POLBKDM4EATMTRPV1ICMT
SCHEMBL9309835 0.82 UNG (0.49) POLBKDM4EATMTRPV1ICMT
SCHEMBL28721627 0.81 ALDH1A1 (0.58) POLBALDH1A1GLATDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0194693-B1 POLYPRENYL COMPOUNDS, PROCESSES FOR PREPARING THEM, AND PHARMACEUTICAL COMPOSITION CONTAINING THEM Eisai Co., Ltd. (JP) 1989-07-26 EP claimed
US-4788330-A Polyprenyl compounds EISAI CO., LTD. (JP) 1988-11-29 US claimed
EP-0194693-A1 Polyprenyl compounds, processes for preparing them, and pharmaceutical composition containing them Eisai Co., Ltd. (JP) 1986-09-17 EP claimed
US-5428028-A Method for lowering cholesterol employing a phosphonomethylphosphinate squalene synthetase inhibitor E. R. SQUIBB & SONS, INC. (US) 1995-06-27 US disclosed
US-5374628-A Aryl and heteroaryl(phosphinylmethyl)phosphonate squalene synthetase inhibitors and method E. R. SQUIBB & SONS, INC. (US) 1994-12-20 US disclosed
US-5278153-A Hypocholesterolemic or hypolipemic E. R. SQUIBB & SONS, INC. (US) 1994-01-11 US disclosed
EP-0513761-A2 Bisphosphonate squalene synthetase inhibitors E.R. SQUIBB & SONS, INC. (US) 1992-11-19 EP disclosed
EP-0514124-A2 Use of phosphonomethylphosphinate squalene synthetase inhibitors for the manufacture of a medicament for the lowering cholesterol E.R. SQUIBB & SONS, INC. (US) 1992-11-19 EP disclosed
US-5157027-A Anticholesterol agents E. R. SQUIBB & SONS, INC. (US) 1992-10-20 US disclosed
US-4883916-A ANTICHOLESTEROL, ANTIARTERIOSCELEROSIS EISAI CO., LTD. (JP) 1989-11-28 US disclosed
EP-0194693-B1 POLYPRENYL COMPOUNDS, PROCESSES FOR PREPARING THEM, AND PHARMACEUTICAL COMPOSITION CONTAINING THEM Eisai Co., Ltd. (JP) 1989-07-26 EP disclosed
US-4788330-A Polyprenyl compounds EISAI CO., LTD. (JP) 1988-11-29 US disclosed
EP-0194693-A1 Polyprenyl compounds, processes for preparing them, and pharmaceutical composition containing them Eisai Co., Ltd. (JP) 1986-09-17 EP disclosed