SCHEMBL9129387

SCHEMBL9129387

OCC1CCCN(C2(c3ccccc3)CCCCC2)C1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.58
GRIN1 Q05586 2/20 0.58
GRIN2A Q12879 2/20 0.58
GRIN2B Q13224 2/20 0.58
GRIN2D O15399 1/20 0.58
GRIN3B O60391 1/20 0.58
CYP2B6 P20813 1/20 0.58
SLC6A2 P23975 1/20 0.58
SLC6A4 P31645 1/20 0.58
PRCP P42785 1/20 0.58
SLC6A3 Q01959 1/20 0.58
KCNH2 Q12809 1/20 0.58
GRIN2C Q14957 1/20 0.58
GRIN3A Q8TCU5 1/20 0.58
OPRM1 P35372 5/20 0.56
OPRD1 P41143 1/20 0.56
MMP2 P08253 1/20 0.49
MMP9 P14780 1/20 0.49
CYP2D6 P10635 1/20 0.45
NPC1 O15118 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5673899 0.83 SLC6A2 (0.54) SIGMAR1GRIN1GRIN2AGRIN2BGRIN2D
SCHEMBL7697741 0.79 KMT2A (0.62) SIGMAR1SLC6A2PRCPOPRM1MMP2
SCHEMBL5674113 0.78 SIGMAR1 (0.63) SIGMAR1GRIN1GRIN2AGRIN2BGRIN2D
SCHEMBL5674111 0.78 SIGMAR1 (0.63) SIGMAR1GRIN1GRIN2AGRIN2BGRIN2D
SCHEMBL9129917 0.78 SIGMAR1 (0.58) SIGMAR1GRIN1GRIN2AGRIN2BGRIN2D
Rolicyclidine SCHEMBL517928 0.75 SIGMAR1 (1.00) SIGMAR1GRIN1GRIN2AGRIN2BGRIN2D
SCHEMBL9153279 0.75 SIGMAR1 (1.00) SIGMAR1GRIN1GRIN2AGRIN2BGRIN2D
SCHEMBL3407261 0.75 GRIN1 (0.92) SIGMAR1GRIN1GRIN2AGRIN2BGRIN2D
Phencyclidine SCHEMBL17008793 0.75 SIGMAR1 (1.00) SIGMAR1GRIN1GRIN2AGRIN2BGRIN2D
Phencyclidine SCHEMBL42022 0.75 SIGMAR1 (1.00) SIGMAR1GRIN1GRIN2AGRIN2BGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459387-B1 Phencyclidine and phencyclidine metabolites assay, tracers, immunogens, antibodies and reagent kit ABBOTT LAB (US) 1995-09-20 EP disclosed
US-5407834-A Monoclonal antibody which binds phencyclidine and metabolites, raised against specified immunogen, lacking specifed cross reactivity ABBOTT LABORATORIES (US) 1995-04-18 US disclosed
US-5155212-A Substituted phencyclidine compound linked to polyamino acid ABBOTT LABORATORIES (US) 1992-10-13 US disclosed
EP-0459387-A2 Phencyclidine and phencyclidine metabolites assay, tracers, immunogens, antibodies and reagent kit ABBOTT LABORATORIES (US) 1991-12-04 EP disclosed