SCHEMBL9130259

SCHEMBL9130259

COc1cc2c(cc1OC)C(CCCN1CCN(c3ccccc3)CC1)(c1ccc(F)cc1)OCC2

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.44
DRD2 P14416 3/20 0.44
DRD3 P35462 3/20 0.44
HTR1A P08908 2/20 0.44
HTR2A P28223 1/20 0.44
HRH1 P35367 1/20 0.44
TMEM97 Q5BJF2 1/20 0.44
DRD4 P21917 2/20 0.42
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9134820 0.95 KDM4E (0.45) DRD2HTR1AHTR2AKDM4E
SCHEMBL9131769 0.89 DRD2 (0.44) SIGMAR1DRD2DRD3HTR1AHTR2A
SCHEMBL11668436 0.88 KMT2A (0.39)
SCHEMBL9129583 0.88 HTR1A (0.51) SIGMAR1DRD2DRD3HTR1AHTR2A
SCHEMBL11674004 0.86 SIGMAR1 (0.42) SIGMAR1DRD2DRD3HTR1ATMEM97
SCHEMBL9133615 0.85 SIGMAR1 (0.47) SIGMAR1DRD2DRD3HTR1AHTR2A
SCHEMBL11072336 0.84 PARP1 (0.42) SIGMAR1HTR1AKDM4E
SCHEMBL10840660 0.83 HTR1A (0.43) SIGMAR1DRD2DRD3HTR1AHTR2A
SCHEMBL10749348 0.83 KDM4E (0.47) DRD2DRD3HTR1AHTR2ADRD4
SCHEMBL11224396 0.79 SLC6A4 (0.41) SIGMAR1DRD3HTR1AHTR2AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992018089-A2 USE OF STEROIDAL AND NON-STEROIDAL AMINES TO SENSITIZE MULTIDRUG-RESISTANT CELLS THE UPJOHN COMPANY (US) 1992-10-29 WO claimed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US claimed
US-5436337-A Anticarcinogenic agents THE UPJOHN COMPANY (US) 1995-07-25 US disclosed
EP-0579754-A1 USE OF AMINES TO SENSITIZE MULTIDRUG-RESISTANT CELLS THE UPJOHN COMPANY (US) 1994-01-26 EP disclosed
WO-1992018089-A2 USE OF STEROIDAL AND NON-STEROIDAL AMINES TO SENSITIZE MULTIDRUG-RESISTANT CELLS THE UPJOHN COMPANY (US) 1992-10-29 WO disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed