SCHEMBL10749348

SCHEMBL10749348

COc1cc2c(cc1OC)C(C)(CCCN1CCN(c3ccc(F)cc3)CC1)OCC2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C19 P33261 1/20 0.45
MAOB P27338 1/20 0.44
DRD2 P14416 2/20 0.42
MAPK1 P28482 1/20 0.41
HTR7 P34969 2/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ABCB1 P08183 2/20 0.41
HTR4 Q13639 1/20 0.41
HTR1A P08908 2/20 0.40
HTR2A P28223 2/20 0.40
PKM P14618 1/20 0.40
HTR2C P28335 1/20 0.40
ADRA2A P08913 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9134820 0.87 KDM4E (0.45) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL9131446 0.84 KDM4E (0.48) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL9130259 0.83 SIGMAR1 (0.44) KDM4EDRD2HTR1AHTR2ADRD4
SCHEMBL11567437 0.82 DRD2 (0.49) CYP1A2CYP2C19DRD2HTR7HTR1A
SCHEMBL10752570 0.80 HTR1A (0.54) MAOBDRD2HTR7HTR1AHTR2A
SCHEMBL11668436 0.77 KMT2A (0.39) ALDH1A1CYP1A2CYP2D6ABCB1
SCHEMBL11567096 0.76 ADORA2A (0.36) DRD2DRD4DRD3
SCHEMBL9130488 0.76 DRD2 (0.46) KDM4EMAPTDRD2MAPK1HTR7
SCHEMBL9131769 0.75 DRD2 (0.44) ALDH1A1MAPTDRD2HTR7LMNA
SCHEMBL10744900 0.74 HTR7 (0.44) KDM4EMAPTHTR7HTR1ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4711960-A HYPOTENSIVE, ANTIPSYCHOTIC AGENTS THE UPJOHN COMPANY (US) 1987-12-08 US disclosed
US-4577021-A PSYCHOLOGICAL DISORDERS, HYPOTENSIVE THE UPJOHN COMPANY (US) 1986-03-18 US disclosed
US-4487774-A Isochromans THE UPJOHN COMPANY (US) 1984-12-11 US disclosed