SCHEMBL9130785

SCHEMBL9130785

O=C1COc2ccc(CC(=O)N3Cc4ccccc4CC3CN3CCCC3)cc2N1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.46
DRD2 P14416 2/20 0.46
DRD4 P21917 2/20 0.46
DRD3 P35462 1/20 0.46
OPRK1 P41145 3/20 0.44
CXCR3 P49682 1/20 0.43
HTR1A P08908 1/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
SLC6A4 P31645 1/20 0.42
NR3C2 P08235 1/20 0.42
CPT2 P23786 1/20 0.41
CPT1A P50416 1/20 0.41
CPT1B Q92523 1/20 0.41
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9128047 0.89 PARP1 (0.47) PARP1DRD2DRD4DRD3OPRK1
SCHEMBL9130335 0.81 OPRD1 (0.64) PARP1DRD2DRD4DRD3OPRK1
SCHEMBL9130908 0.79 OPRK1 (0.48) DRD4OPRK1NPC1
SCHEMBL9129888 0.78 OPRK1 (0.46) DRD4OPRK1NPC1
Hydrochloric Acid SCHEMBL10690631 0.77 OPRK1 (0.67) DRD4OPRK1NPC1
Hydrochloric Acid SCHEMBL9803205 0.77 OPRK1 (0.67) DRD4OPRK1NPC1
Hydrochloric Acid SCHEMBL10691626 0.77 OPRK1 (0.67) DRD4OPRK1NPC1
SCHEMBL9126782 0.76 OPRK1 (0.45) DRD4OPRK1NPC1
SCHEMBL14073049 0.75 PARP1 (0.56) PARP1DRD2DRD4DRD3NR3C2
SCHEMBL14073038 0.72 PARP1 (0.48) PARP1DRD2DRD4DRD3CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1121072-A Acetamides MERCK PATENG GES MIT BESCHRANK (DE) 1996-04-24 CN disclosed
US-5472961-A Acetamides MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-12-05 US disclosed
EP-0670318-A2 Acetamides with analgesic and neuroprotective activity MERCK PATENT GmbH (DE) 1995-09-06 EP disclosed