SCHEMBL9130908

SCHEMBL9130908

O=C(Cc1ccc2[nH]c(=O)[nH]c2c1)N1Cc2ccccc2CC1CN1CCCC1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 7/20 0.48
OPRD1 P41143 3/20 0.44
NPC1 O15118 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
NFKB1 P19838 1/20 0.44
CYP2C19 P33261 1/20 0.44
HIF1A Q16665 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
BLM P54132 1/20 0.44
PMP22 Q01453 1/20 0.44
DRD4 P21917 1/20 0.44
SLC6A3 Q01959 1/20 0.44
TMEM97 Q5BJF2 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
KCNH2 Q12809 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9129660 0.88 OPRK1 (0.48) OPRK1
SCHEMBL9129888 0.85 OPRK1 (0.46) OPRK1OPRD1NPC1CYP1A2CYP3A4
SCHEMBL9126782 0.84 OPRK1 (0.45) OPRK1OPRD1NPC1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9803205 0.82 OPRK1 (0.67) OPRK1OPRD1NPC1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL10690631 0.82 OPRK1 (0.67) OPRK1OPRD1NPC1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL10691626 0.82 OPRK1 (0.67) OPRK1OPRD1NPC1CYP1A2CYP3A4
SCHEMBL9130785 0.79 PARP1 (0.46) OPRK1NPC1DRD4
SCHEMBL9131226 0.79 OPRD1 (0.71) OPRK1OPRD1
SCHEMBL9130848 0.74 OPRK1 (0.45) OPRK1KCNH2
SCHEMBL9129777 0.73 OPRK1 (0.45) OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5472961-A Acetamides MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-12-05 US disclosed
EP-0670318-A2 Acetamides with analgesic and neuroprotective activity MERCK PATENT GmbH (DE) 1995-09-06 EP disclosed