SCHEMBL9136332

SCHEMBL9136332

CCOC(=O)C1(c2cccc(O)c2)CCOCC1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.54
ALDH1A1 P00352 1/20 0.52
OPRM1 P35372 6/20 0.51
LMNA P02545 1/20 0.51
TSHR P16473 1/20 0.51
CYP2C19 P33261 1/20 0.51
OPRD1 P41143 3/20 0.50
OPRK1 P41145 3/20 0.50
SLC22A1 O15245 1/20 0.50
SLC6A4 P31645 1/20 0.50
ADRA1A P35348 1/20 0.50
KCNH2 Q12809 1/20 0.50
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4950745 0.90 OPRM1 (0.57) OPRM1OPRD1OPRK1SLC22A1SLC6A4
SCHEMBL7807438 0.86 ALDH1A1 (0.51) ALOX5ALDH1A1OPRM1LMNATSHR
SCHEMBL27078112 0.85 CYP2C19 (0.45) ALOX5ALDH1A1LMNATSHRCYP2C19
SCHEMBL29731283 0.85 CYP2C19 (0.45) ALOX5ALDH1A1LMNATSHRCYP2C19
Hydroxypethidine SCHEMBL29966554 0.83 OPRM1 (0.74) OPRM1OPRD1OPRK1SLC22A1SLC6A4
SCHEMBL18808528 0.83 OPRM1 (0.50) OPRM1OPRD1OPRK1SLC22A1SLC6A4
Hydroxypethidine SCHEMBL25246 0.83 OPRM1 (0.74) OPRM1OPRD1OPRK1SLC22A1SLC6A4
Hydroxypethidine SCHEMBL317328 0.82 OPRM1 (0.74) OPRM1OPRD1OPRK1SLC22A1SLC6A4
SCHEMBL7810873 0.81 ALOX5 (0.67) ALOX5ALDH1A1OPRM1LMNATSHR
SCHEMBL1600273 0.81 ALOX5 (0.55) ALOX5ALDH1A1OPRM1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462830-B1 Cyclic ether derivatives ZENECA LTD (GB) 1995-10-18 EP disclosed
US-5407945-A Pyran derivatives and their use as inhibitors of 5-lipoxygenase IMPERIAL CHEMICAL INDUSTRIES, INC. (GB) 1995-04-18 US disclosed
US-5254581-A Used in the treatment of various inflammatory and allergic diseases IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-10-19 US disclosed
EP-0462830-A2 Cyclic ether derivatives ZENECA LIMITED (GB) 1991-12-27 EP disclosed