SCHEMBL9137641

SCHEMBL9137641

CCCc1nc(N)c(C(=O)OCC)[nH]1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.65
KDM4E B2RXH2 5/20 0.65
HPGD P15428 3/20 0.65
HTT P42858 1/20 0.65
RECQL P46063 1/20 0.65
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HSP90AA1 P07900 1/20 0.43
GAA P10253 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 2/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9206394 0.91 ALDH1A1 (0.61) ALDH1A1KDM4EHPGDHTTRECQL
SCHEMBL9199916 0.86 HPGD (0.46) ALDH1A1KDM4EHPGDHTTRECQL
SCHEMBL4356883 0.84 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDHTTRECQL
SCHEMBL5809049 0.84 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDHTTRECQL
SCHEMBL1275935 0.83 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHTTRECQL
Hydrochloric Acid SCHEMBL1417761 0.81 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDHTTRECQL
SCHEMBL7234563 0.80 ALDH1A1 (0.39) ALDH1A1KDM4EHPGDHTTRECQL
SCHEMBL27609241 0.80 ALDH1A1 (0.39) ALDH1A1KDM4EHPGDHTTRECQL
SCHEMBL1444895 0.80 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDHTTRECQL
SCHEMBL8664938 0.80 KDM4E (0.50) ALDH1A1KDM4EHPGDHTTRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5389661-A Treats hypertension, heart failure, glaucoma and hyperaldosteronism WARNER-LAMBERT COMPANY (US) 1995-02-14 US disclosed
US-5322950-A Treating hypertension, hyperaldosteronism, glaucoma, heart failure WARNER-LAMBERT COMPANY (US) 1994-06-21 US disclosed