SCHEMBL9145488

SCHEMBL9145488

CC1(C)CN(C2=CCCC2=O)c2cc(Br)ccc2O1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.38
CTSD P07339 1/20 0.38
PIK3CD O00329 3/20 0.36
PIK3CA P42336 3/20 0.36
PIK3CB P42338 3/20 0.36
PIK3CG P48736 3/20 0.36
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
PKM P14618 1/20 0.33
NPR1 P16066 1/20 0.33
TSHR P16473 1/20 0.33
BLM P54132 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MALT1 Q9UDY8 1/20 0.33
MAOB P27338 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 1/20 0.32
PBRM1 Q86U86 1/20 0.32
PDE3B Q13370 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9146876 0.83 CTSD (0.35) BACE1CTSDMALT1ALDH1A1SRD5A1
SCHEMBL9147914 0.83 PARP1 (0.34) TP53MAPTSRD5A1
SCHEMBL9146937 0.82 ABCC9 (0.36) BACE1CTSDCYP1A2MALT1MAOB
SCHEMBL9143553 0.76 ABCC9 (0.37) BACE1CTSDCYP1A2MALT1MAOB
SCHEMBL9147151 0.75 CASP6 (0.38) TDP1MALT1ALDH1A1MAPTNR3C2
SCHEMBL27321636 0.69 KMT2A (0.40) BACE1CTSDPIK3CDPIK3CAPIK3CB
SCHEMBL9146574 0.68 BACE1 (0.35) BACE1CTSDPIK3CDPIK3CAPIK3CB
SCHEMBL9147618 0.66 BACE1 (0.35) BACE1CTSDTP53TSHRALDH1A1
SCHEMBL9146857 0.65 ABCC9 (0.30) CYP1A2LMNA
SCHEMBL9146859 0.65 ABCC9 (0.30) CYP1A2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5420126-A Potassium channel activators YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0432893-A2 Benzoxazine derivatives, their preparation and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1991-06-19 EP disclosed