SCHEMBL9152657

SCHEMBL9152657

CON(C)C(=O)c1ccc(-c2ccc(C)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.53
TDP1 Q9NUW8 2/20 0.47
ALDH1A1 P00352 9/20 0.43
LMNA P02545 4/20 0.43
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
HSD17B2 P37059 4/20 0.43
HSD17B1 P14061 3/20 0.43
SMN1; SMN2 Q16637 4/20 0.42
HPGD P15428 4/20 0.40
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
CDK2 P24941 1/20 0.40
TP53 P04637 1/20 0.40
HTT P42858 3/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 2/20 0.39
ATM Q13315 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL870352 0.94 MLYCD (0.57) MLYCDTDP1ALDH1A1LMNACES2
SCHEMBL9707103 0.86 MLYCD (0.54) MLYCDTDP1ALDH1A1LMNACES2
SCHEMBL4449884 0.85 MAPT (0.56) MLYCDALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL8816853 0.84 HDAC1 (0.54) MLYCDALDH1A1SMN1; SMN2HPGDHTT
SCHEMBL13670740 0.84 MEN1 (0.51) MLYCDTDP1ALDH1A1LMNACES2
SCHEMBL5209405 0.81 HDAC1 (0.46) ATM
SCHEMBL8312870 0.81 MLYCD (0.49) MLYCDTDP1ALDH1A1HSD17B2SMN1; SMN2
SCHEMBL16574187 0.80 ALDH1A1 (0.55) TDP1ALDH1A1LMNACES2CES1
SCHEMBL9154730 0.80 MLYCD (0.48) MLYCDALDH1A1CES2CES1HSD17B2
SCHEMBL8046453 0.80 HRH3 (0.55) MLYCDHSD17B2HSD17B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0464465-B1 Substituted aminoalkylbiphenyl derivatives, antimycotic composition containing them, and intermediates for their preparation HOFFMANN LA ROCHE (CH) 1995-01-11 EP disclosed
US-5239084-A Chmical intermeidates for fungicides, mycosis HOFFMANN-LA ROCHE INC. (US) 1993-08-24 US disclosed
US-5177067-A Fungicides HOFFMANN-LAROCHE INC. (US) 1993-01-05 US disclosed
EP-0464465-A1 Substituted aminoalkylbiphenyl derivatives, antimycotic composition containing them, and intermediates for their preparation F. HOFFMANN-LA ROCHE AG (CH) 1992-01-08 EP disclosed