SCHEMBL9155180

SCHEMBL9155180

CN(CCCCNC(=O)C/C=C/c1ccc(-n2ccc(=O)cc2)cc1)CCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.42
TMEM97 Q5BJF2 1/20 0.42
HDAC1 Q13547 2/20 0.39
HDAC2 Q92769 2/20 0.39
HDAC8 Q9BY41 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9160658 0.87 CNR1 (0.36)
SCHEMBL9158516 0.87 TBXAS1 (0.41) SIGMAR1TMEM97
SCHEMBL9232408 0.86 CYP3A4 (0.42) SIGMAR1TMEM97ALDH1A1
SCHEMBL9160168 0.84 CYP3A4 (0.40) SIGMAR1TMEM97ALDH1A1
SCHEMBL9232815 0.84 CNR1 (0.36) SIGMAR1LMNA
SCHEMBL8828152 0.84 TMEM97 (0.43) SIGMAR1TMEM97
SCHEMBL9160871 0.84 CCR3 (0.36) SIGMAR1TMEM97HDAC1HDAC6
SCHEMBL8828169 0.83 OPRM1 (0.44) SIGMAR1TMEM97ALDH1A1
SCHEMBL9156723 0.79 MAOB (0.46) ALDH1A1LMNA
SCHEMBL9159739 0.78 MAOB (0.42) SIGMAR1TMEM97ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430059-A Treating heart disease EISAI CO., LTD. (JP) 1995-07-04 US disclosed
EP-0633248-A1 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1995-01-11 EP disclosed
EP-0589491-A1 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1994-03-30 EP disclosed
US-5292770-A Butenoic acid derivatives EISAI CO., LTD. (JP) 1994-03-08 US disclosed
US-5166188-A Cardiovascular disorders, antiischemic agents EISAI CO., LTD. (JP) 1992-11-24 US disclosed
EP-0399358-A2 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1990-11-28 EP disclosed