SCHEMBL9156987

SCHEMBL9156987

COc1ccc(CN2CCN(C(=O)[C@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c(OC)c1OC

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
HTT P42858 1/20 0.55
CYP2C19 P33261 2/20 0.52
MEN1 O00255 5/20 0.51
KMT2A Q03164 5/20 0.51
KDM4E B2RXH2 1/20 0.51
PKM P14618 1/20 0.51
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
P2RX7 Q99572 6/20 0.49
ALOX15 P16050 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.46
P2RY12 Q9H244 1/20 0.46
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
HCRTR2 O43614 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9426160 0.99 ALDH1A1 (0.55) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9426873 0.94 ITGB3 (0.51) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9426241 0.93 MEN1 (0.49) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9158857 0.92 P2RX7 (0.53) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9426464 0.92 ALDH1A1 (0.55) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9426250 0.91 ALDH1A1 (0.53) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9154136 0.89 CYP2C19 (0.56) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9154447 0.89 CYP2C19 (0.56) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9154438 0.89 ALDH1A1 (0.51) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9425893 0.89 ALDH1A1 (0.51) ALDH1A1HTTCYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533516-B1 Amides of 1-(alkoxybenzyl)piperazines, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 1995-02-08 EP disclosed
US-5340809-A Antihypoxic, antiischemic agents ADIR ET COMPAGNIE (FR) 1994-08-23 US disclosed
EP-0533516-A2 Amides of 1-(alkoxybenzyl)piperazines, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1993-03-24 EP disclosed