SCHEMBL9163375

SCHEMBL9163375

Nc1cnc2ccc(SC(F)F)cc2c1-c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 2/20 0.36
MAP4K4 O95819 1/20 0.35
TLR9 Q9NR96 1/20 0.34
LMNA P02545 3/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
STAT3 P40763 1/20 0.32
MAPK10 P53779 1/20 0.32
ATM Q13315 2/20 0.32
KDM4E B2RXH2 2/20 0.32
ACHE P22303 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9159524 0.82 DHODH (0.41) METMAP4K4TLR9LMNAMAPT
SCHEMBL9167207 0.79 MEN1 (0.37) NPC1MAPTRAB9AALDH1A1MEN1
SCHEMBL9164976 0.76 MAP4K4 (0.41) METMAP4K4MAPTALDH1A1CYP1A2
SCHEMBL9161172 0.75 ALDH1A1 (0.52) LMNANPC1MAPTRAB9ASMN1; SMN2
SCHEMBL9164616 0.74 ATM (0.40) METMAP4K4TLR9NPC1RAB9A
SCHEMBL9169732 0.74 ESR1 (0.47) METMAPTALDH1A1KDM4EMEN1
Ammonia Solution, Strong SCHEMBL2249468 0.73 ALDH1A1 (0.51) LMNANPC1MAPTRAB9ASMN1; SMN2
SCHEMBL18057691 0.73 NCF1 (0.47) MAPTSMN1; SMN2NPSR1ALDH1A1CYP1A2
SCHEMBL9164642 0.71
SCHEMBL9163362 0.71 MAPT (0.52) METMAP4K4LMNANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0354994-B1 Quinoline derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-01-25 EP disclosed
US-5254565-A Enzyme inhibitors; anticholesterol agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-19 US disclosed
EP-0354994-A2 Quinoline derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-02-21 EP disclosed