SCHEMBL9164976

SCHEMBL9164976

Nc1cnc2ccc(OC(F)F)cc2c1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.41
GRM2 Q14416 1/20 0.41
DPP4 P27487 6/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
HPGD P15428 2/20 0.37
CYP2C19 P33261 2/20 0.37
HTT P42858 1/20 0.37
HDAC4 P56524 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MET P08581 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9159566 0.79 EIF4E (0.40) GRM2ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL9163375 0.76 MET (0.36) MAP4K4ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL9161172 0.75 ALDH1A1 (0.52) ALDH1A1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL9164616 0.74 ATM (0.40) MAP4K4DPP4ALDH1A1HTTMET
SCHEMBL9169732 0.74 ESR1 (0.47) ALDH1A1KDM4EMAPTMET
Ammonia Solution, Strong SCHEMBL2249468 0.73 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL18057691 0.73 NCF1 (0.47) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9163362 0.71 MAPT (0.52) MAP4K4ALDH1A1HPGDHTTKDM4E
SCHEMBL9159524 0.71 DHODH (0.41) MAP4K4ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL30513838 0.70 MAP4K4 (0.54) MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1028754-C process for preparing quinoline derivatives TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-06-07 CN disclosed
EP-0354994-B1 Quinoline derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-01-25 EP disclosed
US-5254565-A Enzyme inhibitors; anticholesterol agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-19 US disclosed
EP-0354994-A2 Quinoline derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-02-21 EP disclosed
CN-1039416-A Quinoline and preparation thereof and purposes TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1990-02-07 CN disclosed