SCHEMBL9169732

SCHEMBL9169732

Nc1cnc2ccc(C(F)(F)F)cc2c1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.47
MET P08581 1/20 0.45
NPBWR1 P48145 1/20 0.43
TACR1 P25103 2/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
FABP4 P15090 2/20 0.42
FABP5 Q01469 2/20 0.42
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
DGAT1 O75907 1/20 0.41
KCNH2 Q12809 1/20 0.41
DHODH Q02127 1/20 0.41
KIF11 P52732 1/20 0.40
ABCG2 Q9UNQ0 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29742208 0.79 BACE1 (0.45) NPBWR1CCNCCDK8KDM4EALDH1A1
SCHEMBL23935164 0.79 BACE1 (0.45) NPBWR1CCNCCDK8KDM4EALDH1A1
SCHEMBL9161172 0.78 ALDH1A1 (0.52) ESR1FABP4FABP5KDM4EALDH1A1
SCHEMBL9162858 0.78 ABCG2 (0.43) ESR1TACR1DHODHABCG2MEN1
SCHEMBL29712652 0.77 GRM5 (0.46) ESR1KDM4EALDH1A1MAPT
SCHEMBL28328975 0.77 GRM5 (0.46) ESR1KDM4EALDH1A1MAPT
Ammonia Solution, Strong SCHEMBL2249468 0.77 ALDH1A1 (0.51) ESR1FABP4FABP5KDM4EALDH1A1
SCHEMBL18057691 0.76 NCF1 (0.47) ESR1ADORA2AKCNH2KDM4EMEN1
SCHEMBL23747858 0.75 NR1H2 (0.41) ESR1NPBWR1TACR1FABP4FABP5
SCHEMBL9159524 0.74 DHODH (0.41) METDHODHABCG2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0354994-B1 Quinoline derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-01-25 EP disclosed
US-5254565-A Enzyme inhibitors; anticholesterol agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-19 US disclosed
EP-0354994-A2 Quinoline derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-02-21 EP disclosed