Niacinamide

Niacinamide

SCHEMBL9164048

Cc1nc(Cl)nc2nc[nH]c12.NC(=O)c1cccnc1

nearest known ligand 0.50

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F7 P08709 1/20 0.50
F3 P13726 1/20 0.50
SARM1 Q6SZW1 1/20 0.50
SIRT2 Q8IXJ6 1/20 0.50
SIRT6 Q8N6T7 1/20 0.50
SIRT1 Q96EB6 1/20 0.50
SIRT3 Q9NTG7 1/20 0.50
SIRT5 Q9NXA8 1/20 0.50
SIRT4 Q9Y6E7 1/20 0.50
NEK2 P51955 2/20 0.40
MKNK1 Q9BUB5 4/20 0.39
MKNK2 Q9HBH9 3/20 0.39
XDH P47989 1/20 0.39
F2 P00734 2/20 0.38
HSD17B10 Q99714 1/20 0.38
TSHR P16473 1/20 0.38
PIK3CA P42336 1/20 0.37
PIK3CG P48736 1/20 0.37
CHRM4 P08173 1/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Niacinamide SCHEMBL9164041 0.82 F7 (0.50) F7F3SARM1SIRT2SIRT6
Hypoxanthine SCHEMBL472854 0.78 F7 (0.61) F7F3SARM1SIRT2SIRT6
Guanine SCHEMBL1266684 0.76 PNP (0.60) F7F3SARM1SIRT2SIRT6
Mercaptopurine Anhydrous SCHEMBL6558420 0.76 F7 (0.58) F7F3SARM1SIRT2SIRT6
SCHEMBL4451634 0.75 XDH (0.61) XDH
Niacinamide SCHEMBL4731742 0.75 F7 (0.54) F7F3SARM1SIRT2SIRT6
Thioguanine SCHEMBL2314990 0.75 F7 (0.50) F7F3SARM1SIRT2SIRT6
Adenine SCHEMBL9274699 0.74 PI4KA (0.52) F7F3SARM1SIRT2SIRT6
Adenine SCHEMBL22748487 0.74 PI4KA (0.55) F7F3SARM1SIRT2SIRT6
Adenine SCHEMBL2564210 0.74 PI4KA (0.55) F7F3SARM1SIRT2SIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470201-B1 METHOD OF ANALYSIS, REAGENT COMPOSITION AND USE THEREOF FOR GLUCOSE DETERMINATION MIGRATA UK LTD (GB) 1995-05-03 EP claimed
EP-0470201-A1 METHOD OF ANALYSIS, REAGENT COMPOSITION AND USE THEREOF FOR GLUCOSE DETERMINATION. MIGRATA UK LTD (GB) 1992-02-12 EP claimed
WO-1990012889-A1 METHOD OF ANALYSIS, REAGENT COMPOSITION AND USE THEREOF FOR GLUCOSE DETERMINATION MIGRATA UK LTD (GB) 1990-11-01 WO claimed
EP-0470201-B1 METHOD OF ANALYSIS, REAGENT COMPOSITION AND USE THEREOF FOR GLUCOSE DETERMINATION MIGRATA UK LTD (GB) 1995-05-03 EP disclosed
US-5278047-A Quantitative determination by spectrophotometry LILJA JAN E (SE) 1994-01-11 US disclosed
EP-0470201-A1 METHOD OF ANALYSIS, REAGENT COMPOSITION AND USE THEREOF FOR GLUCOSE DETERMINATION. MIGRATA UK LTD (GB) 1992-02-12 EP disclosed
WO-1990012889-A1 METHOD OF ANALYSIS, REAGENT COMPOSITION AND USE THEREOF FOR GLUCOSE DETERMINATION MIGRATA UK LTD (GB) 1990-11-01 WO disclosed