SCHEMBL9164487

SCHEMBL9164487

CC=CCC(C(=O)O)C(=O)c1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLOD2 O00469 1/20 0.49
ALDH1A1 P00352 3/20 0.47
APP P05067 1/20 0.47
GAA P10253 1/20 0.47
HCAR3 P49019 1/20 0.47
HCAR2 Q8TDS4 1/20 0.47
TBXAS1 P24557 11/20 0.45
GPR52 Q9Y2T5 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
F7 P08709 1/20 0.42
F3 P13726 1/20 0.42
SARM1 Q6SZW1 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
SIRT6 Q8N6T7 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
SIRT3 Q9NTG7 1/20 0.42
SIRT5 Q9NXA8 1/20 0.42
SIRT4 Q9Y6E7 1/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9765887 0.82 TBXAS1 (0.54) PLOD2ALDH1A1APPGAAHCAR3
SCHEMBL9164237 0.82 CYP1A2 (0.42) PLOD2ALDH1A1GPR52L3MBTL1LMNA
SCHEMBL5162022 0.80 ALDH1A1 (0.55) PLOD2ALDH1A1APPGAAHCAR3
SCHEMBL2228198 0.76 ALDH1A1 (0.46) PLOD2ALDH1A1APPGAAHCAR3
SCHEMBL23926879 0.75 L3MBTL1 (0.54) PLOD2ALDH1A1APPGAAHCAR3
SCHEMBL6900351 0.75 ALDH1A1 (0.51) PLOD2ALDH1A1APPGAAHCAR3
SCHEMBL6511843 0.75 MDM2 (0.62) PLOD2ALDH1A1APPGAAHCAR3
SCHEMBL27623816 0.74 TBXAS1 (0.57) TBXAS1TBXA2R
SCHEMBL13898363 0.74 MDM2 (0.47) ALDH1A1L3MBTL1LMNACYP3A4TDP1
SCHEMBL82140 0.73 ALDH1A1 (0.58) PLOD2ALDH1A1APPGAAHCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1040753-C Pyridine derivatives and the preparation thereof ICI PLC (GB) 1998-11-18 CN disclosed
US-5401849-A FOR ANTAGONIZING THE ACTIONS OF, AND INHIBITING THE SYNTHESIS OF, THROMBOXANE A2 ZENECA LIMITED (GB) 1995-03-28 US disclosed
EP-0329360-B1 Pyridine derivatives ICI PLC (GB) 1994-08-03 EP disclosed
US-5248780-A Thromboxane inhibitors IMPERIAL CHEMICAL INDUSTRIES, PLC (GB) 1993-09-28 US disclosed
US-5166213-A Antiischemic agents, cardiovascular disorders, antiasthmatics or antiinflammatory agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-11-24 US disclosed
CN-1035115-A Pyridine derivate and preparation method thereof ICI PLC (GB) 1989-08-30 CN disclosed
EP-0329360-A2 Pyridine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-08-23 EP disclosed