SCHEMBL9164572

SCHEMBL9164572

O=CCCC=Cc1ccccc1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.55
CCND1 P24385 1/20 0.55
TRIM24 O15164 1/20 0.52
TRIM33 Q9UPN9 1/20 0.52
NFKB1 P19838 2/20 0.50
JUN P05412 1/20 0.50
NFE2L2 Q16236 1/20 0.50
CA2 P00918 2/20 0.48
CA1 P00915 1/20 0.48
CA4 P22748 1/20 0.48
MAPT P10636 3/20 0.47
LMNA P02545 1/20 0.47
TRPA1 O75762 1/20 0.47
BCHE P06276 1/20 0.44
GUSB P08236 1/20 0.44
APP P05067 2/20 0.42
KDM4E B2RXH2 2/20 0.41
CA12 O43570 1/20 0.41
CHRNA7 P36544 3/20 0.41
AR P10275 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11189518 0.84 CDK4 (0.59) CDK4CCND1TRIM24TRIM33NFKB1
SCHEMBL4453048 0.81 TRPA1 (0.47) CDK4CCND1TRIM24TRIM33NFKB1
SCHEMBL3415700 0.78 CA2 (0.50) CDK4CCND1TRIM24TRIM33NFKB1
SCHEMBL3415698 0.78 CA2 (0.50) CDK4CCND1TRIM24TRIM33NFKB1
SCHEMBL347703 0.78 TRPA1 (0.48) CDK4CCND1TRIM24TRIM33NFKB1
SCHEMBL30337793 0.78 CA2 (0.50) CDK4CCND1TRIM24TRIM33NFKB1
SCHEMBL9164566 0.78 NFKB1 (0.47) CDK4CCND1TRIM24TRIM33NFKB1
SCHEMBL9164563 0.78 NFKB1 (0.47) CDK4CCND1TRIM24TRIM33NFKB1
SCHEMBL9574440 0.78 NFKB1 (0.55) CDK4CCND1TRIM24TRIM33NFKB1
SCHEMBL348173 0.76 TRPA1 (0.46) CDK4CCND1TRIM24TRIM33NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108530427-A A kind of 1,4- pentadiene -3- ketoxime ethers derivative, preparation method and application containing quinazoline 贵州大学 2018-09-14 CN disclosed
CN-1038586-C Pyrazine derivatives and process for preparing same OTSUKA PHARMA CO LTD (JP) 1998-06-03 CN disclosed
US-5459142-A Autoimmune disease, atherosclerosis, antiischemic agents and nephritis OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-10-17 US disclosed
EP-0511879-B1 Pyrazine derivatives OTSUKA PHARMA CO LTD (JP) 1995-03-22 EP disclosed
EP-0511879-A1 Pyrazine derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-04 EP disclosed