SCHEMBL9167645

SCHEMBL9167645

CCCCCCCCCCCCCCCCCCOc1cc(O)cc(C(=O)OCc2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 4/20 0.53
PLA2G2A P14555 1/20 0.53
TDP1 Q9NUW8 2/20 0.52
TSHR P16473 2/20 0.52
ALDH1A1 P00352 1/20 0.52
CYP3A4 P08684 1/20 0.52
MAPK1 P28482 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
CNR1 P21554 1/20 0.52
LMNA P02545 1/20 0.49
SLC6A2 P23975 1/20 0.49
SLC6A3 Q01959 1/20 0.49
KMT2A Q03164 1/20 0.49
ESR1 P03372 3/20 0.48
AKR1C4 P17516 1/20 0.48
AKR1C3 P42330 1/20 0.48
AKR1C2 P52895 1/20 0.48
AKR1C1 Q04828 1/20 0.48
TP53 P04637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9166914 0.90 PLA2G2A (0.57) PLA2G2ATDP1TSHRALDH1A1CYP3A4
SCHEMBL9323915 0.89 PLA2G2A (0.56) PLA2G2ATDP1TSHRALDH1A1CYP3A4
SCHEMBL9162948 0.88 PLA2G2A (0.54) CNR2PLA2G2ATDP1TSHRALDH1A1
SCHEMBL9324895 0.88 PLA2G2A (0.51) PLA2G2ATDP1TSHRALDH1A1CYP3A4
SCHEMBL30036044 0.87 PLA2G2A (0.53) CNR2PLA2G2ATDP1TSHRALDH1A1
SCHEMBL9402583 0.86 PLA2G2A (0.52) CNR2PLA2G2ATDP1TSHRALDH1A1
SCHEMBL9325282 0.86 PLA2G2A (0.52) CNR2PLA2G2ATDP1TSHRALDH1A1
SCHEMBL9402649 0.85 PLA2G2A (0.51) CNR2PLA2G2ATDP1TSHRALDH1A1
SCHEMBL9169597 0.85 PLA2G2A (0.51) CNR2PLA2G2ATDP1TSHRALDH1A1
SCHEMBL21924267 0.85 KMT2A (0.54) TDP1ALDH1A1L3MBTL1LMNASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5446189-A Diester intermediates for diacid enzyme inhibitor HOFFMANN-LA ROCHE INC. (US) 1995-08-29 US disclosed
US-5374772-A Skin disorders, antiinflammatory agents, cardiovascular disorders HOFFMANN-LAROCHE INC. (US) 1994-12-20 US disclosed
US-5324747-A Treatment of inflammatory diseases HOFFMANN-LA ROCHE INC. (US) 1994-06-28 US disclosed
EP-0601385-A1 Disubstituted benzoic acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1994-06-15 EP disclosed
US-5298652-A N-substituted glycines, inhibitors of phospholipase A2 HOFFMANN-LA ROCHE INC. (US) 1994-03-29 US disclosed
EP-0579066-A2 N-substituted anilines F. HOFFMANN-LA ROCHE AG (CH) 1994-01-19 EP disclosed