Bromide

Bromide

SCHEMBL9171973

Br.CCC(C)Nc1cc(O)ccc1O

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 2/20 0.35
ADRA1A known ✓ P35348 2/20 0.35
SLC6A3 known ✓ Q01959 2/20 0.35
ADRB2 known ✓ P07550 1/20 0.35
ADRB1 known ✓ P08588 1/20 0.35
ADRA2A known ✓ P08913 1/20 0.35
ADRA2B known ✓ P18089 1/20 0.35
ADRA2C known ✓ P18825 1/20 0.35
ADRA1D known ✓ P25100 1/20 0.35
SLC6A4 known ✓ P31645 1/20 0.35
HTR3A known ✓ P46098 1/20 0.35
SIGMAR1 known ✓ Q99720 1/20 0.35
CHRM2 known ✓ P08172 1/20 0.34
CYP3A4 P08684 5/20 0.44
HSD17B10 Q99714 4/20 0.44
TSHR P16473 3/20 0.44
HIF1A Q16665 3/20 0.44
ALDH1A1 P00352 3/20 0.44
ALOX15 P16050 3/20 0.44
HSP90AA1 P07900 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28539633 0.79 ALDH1A1 (0.41) CYP3A4HSD17B10TSHRHIF1AALDH1A1
SCHEMBL29441552 0.78 RORC (0.57) CYP3A4HSD17B10TSHRHIF1AALDH1A1
SCHEMBL4213149 0.78 RORC (0.57) CYP3A4HSD17B10TSHRHIF1AALDH1A1
SCHEMBL4229462 0.76 TSHR (0.48) CYP3A4HSD17B10TSHRHIF1AALDH1A1
SCHEMBL5324416 0.71 ALDH1A1 (0.41) HSD17B10TSHRALDH1A1ALOX15TP53
SCHEMBL5324420 0.71 ALDH1A1 (0.41) HSD17B10TSHRALDH1A1ALOX15TP53
SCHEMBL11991459 0.71 CA12 (0.53) HSD17B10ALDH1A1HCAR3LMNAGAA
SCHEMBL3720674 0.71 ALOX15 (0.78) CYP3A4HSD17B10TSHRHIF1AALDH1A1
Bromide SCHEMBL11513468 0.70 IDO1 (0.43) CYP3A4HSD17B10TSHRHIF1AALDH1A1
SCHEMBL8085472 0.69 ALDH1A1 (0.55) CYP3A4HSD17B10TSHRHIF1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0474402-B1 Chromophore-containing compounds for opto-electronic applications ICI PLC (GB) 1995-05-24 EP disclosed
US-5290630-A Chromophore-containing compounds for opto-electronic applications IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-03-01 US disclosed
EP-0474402-A2 Chromophore-containing compounds for opto-electronic applications IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-03-11 EP disclosed