SCHEMBL9175477

SCHEMBL9175477

CCC1=Nc2ccc(N(C)C)cc2C(=O)C1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
PSMB5 P28074 2/20 0.36
CYP3A4 P08684 1/20 0.32
HPGD P15428 1/20 0.32
HIF1A Q16665 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TERT O14746 1/20 0.32
APP P05067 1/20 0.32
ELANE P08246 2/20 0.32
IP6K1 Q92551 1/20 0.31
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9183312 0.77 PDE3B (0.46) ALDH1A1HPGDHIF1AKDM4EPDE3B
SCHEMBL9182853 0.75 CASP3 (0.36)
SCHEMBL9178650 0.75 PARP1 (0.35)
SCHEMBL4764684 0.74 SHMT2 (0.39) ALDH1A1HPGDHIF1ATDP1KDM4E
SCHEMBL9175673 0.73 BRD4 (0.35) ALDH1A1HPGDHSD17B10KDM4EPDE3B
SCHEMBL339090 0.72 ESR1 (0.39) ALDH1A1APP
SCHEMBL340495 0.71 NPSR1 (0.46) ALDH1A1HPGDHSD17B10TDP1KDM4E
SCHEMBL9180722 0.71 KMT2A (0.40) ALDH1A1HPGDKDM4EELANE
SCHEMBL9180961 0.70 ALDH1A1 (0.36) ALDH1A1KDM4E
SCHEMBL1888235 0.70 ALDH1A1 (0.42) ALDH1A1PSMB5CYP3A4HPGDHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5444071-A Hypotensive agent IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-08-22 US disclosed
EP-0412848-B1 Quinoline derivatives, process for their preparation and their use as medicaments ICI PLC (GB) 1995-01-18 EP disclosed
CN-1050187-A New quinoline compound and preparation method thereof ICI PLC (GB) 1991-03-27 CN disclosed
EP-0412848-A2 Quinoline derivatives, process for their preparation and their use as medicaments ZENECA LIMITED (GB) 1991-02-13 EP disclosed