SCHEMBL9182091

SCHEMBL9182091

CCC1=Nc2cc(C#N)ccc2C(=O)C1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 1/20 0.36
CYP2A6 P11509 1/20 0.35
RXRA P19793 4/20 0.33
PGR P06401 1/20 0.33
CASP3 P42574 1/20 0.33
IDO1 P14902 1/20 0.33
MAOB P27338 3/20 0.32
MAOA P21397 2/20 0.32
MALT1 Q9UDY8 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
CYP11B2 P19099 3/20 0.32
CYP11B1 P15538 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9182853 0.89 CASP3 (0.36) EGLN2CYP2A6RXRACASP3MALT1
SCHEMBL9180722 0.79 KMT2A (0.40) MAOBMAOA
SCHEMBL9182860 0.78 HPGD (0.36)
SCHEMBL23920288 0.76 CYP2A6 (0.39) CYP2A6HTR2AHTR2CHTR2BCYP11B2
SCHEMBL9179384 0.75 KDM4E (0.42) MAOB
SCHEMBL4764684 0.73 SHMT2 (0.39) CASP3IDO1MAOBMAOA
SCHEMBL29141181 0.69 CASP3 (0.43) PGRCASP3MAOBMAOAMALT1
SCHEMBL30711519 0.69 CASP3 (0.43) PGRCASP3MAOBMAOAMALT1
SCHEMBL9180114 0.69 CASP3 (0.39) EGLN2CYP2A6CASP3MALT1HTR2A
SCHEMBL9178830 0.69 KDM4E (0.40) HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5444071-A Hypotensive agent IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-08-22 US disclosed
EP-0412848-B1 Quinoline derivatives, process for their preparation and their use as medicaments ICI PLC (GB) 1995-01-18 EP disclosed
EP-0412848-A2 Quinoline derivatives, process for their preparation and their use as medicaments ZENECA LIMITED (GB) 1991-02-13 EP disclosed