SCHEMBL23920288

SCHEMBL23920288

CCC1=Nc2ccc(C#N)cc2C1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.39
DRD2 P14416 4/20 0.37
DRD3 P35462 4/20 0.37
TRPA1 O75762 1/20 0.36
PNMT P11086 4/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
NAMPT P43490 1/20 0.34
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
CYP11B2 P19099 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9182853 0.79 CASP3 (0.36) CYP2A6NOS3NOS1NOS2HTR2A
SCHEMBL23920265 0.76 PDE3B (0.38) NOS3NOS1NOS2HTR2C
SCHEMBL9182091 0.76 EGLN2 (0.36) CYP2A6HTR2AHTR2CHTR2BCYP11B2
SCHEMBL7418032 0.65 NOS2 (0.41) DRD2DRD3TRPA1PNMTNOS3
SCHEMBL6739755 0.64
SCHEMBL7647780 0.63 PNMT (0.44) DRD2DRD3TRPA1PNMTNOS3
SCHEMBL11908201 0.63 PNMT (0.41) DRD2DRD3TRPA1PNMTNOS3
SCHEMBL11017385 0.63 TRPA1 (0.44) DRD2DRD3TRPA1PNMTNOS3
Water SCHEMBL28095232 0.63 PNMT (0.49) DRD2DRD3TRPA1PNMTNOS3
Bromide SCHEMBL17202846 0.63 PNMT (0.52) CYP2A6DRD2DRD3TRPA1PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3892623-A1 COMPOUNDS HAVING PDE9A INHIBITORY ACTIVITY, AND PHARMACEUTICAL USES THEREOF Korea Research Institute of Chemical Technology (KR) 2021-10-13 EP disclosed