SCHEMBL9182128

SCHEMBL9182128

CCOC(=O)CN(C)C(=O)c1cc(C)c(C)cc1C(=O)c1ccccc1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
ALDH1A1 P00352 3/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
GAA P10253 1/20 0.40
TSHR P16473 2/20 0.40
KCNK3 O14649 1/20 0.39
MAPK13 O15264 2/20 0.39
MAPK12 P53778 2/20 0.39
MAPK11 Q15759 2/20 0.39
MAPK14 Q16539 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7850510 0.84 KMT2A (0.39) KMT2AMEN1CA12CA1CA2
SCHEMBL7374457 0.80 TACR1 (0.51) KMT2AMEN1CA12CA1CA2
SCHEMBL8785404 0.76 KMT2A (0.47) KMT2AALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL13468195 0.75 KMT2A (0.58) KMT2AMEN1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL8785261 0.74 LMNA (0.46) KMT2AMEN1CA12CA1CA2
SCHEMBL7374463 0.73 ALDH1A1 (0.50) KMT2AMEN1CA12CA1CA2
SCHEMBL7849671 0.72 ALDH1A1 (0.52) KMT2AMEN1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL12499605 0.72 KMT2A (0.43) KMT2AMEN1RAB9ASMN1; SMN2NPC1
SCHEMBL7375054 0.72 PDE3B (0.49) KMT2AMEN1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL9401553 0.72 LMNA (0.43) CA12CA1CA2CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481383-B1 Heterocyclic amine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-06-28 EP disclosed
US-5300646-A Intermediates for acylcoenzyme A:cholesterol acyltransferase inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-04-05 US disclosed
US-5198462-A Acyl Coenzyme A:Cholesterol Transferase Inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-03-30 US disclosed
EP-0481383-A1 Heterocyclic amine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1992-04-22 EP disclosed