SCHEMBL9185477

SCHEMBL9185477

COc1ccc(C(O)C(Cl)C(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.47
AKR1C3 P42330 6/20 0.46
AKR1C2 P52895 6/20 0.46
PTGS2 P35354 3/20 0.46
PTGS1 P23219 3/20 0.46
CYP1A2 P05177 2/20 0.46
TSHR P16473 2/20 0.46
CDC42 P60953 1/20 0.46
RAC1 P63000 1/20 0.46
SLC22A6 Q4U2R8 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
ACP3 P15309 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
ALDH1A1 P00352 2/20 0.44
GRM8 O00222 1/20 0.43
GRM6 O15303 1/20 0.43
GRM4 Q14833 1/20 0.43
NPSR1 Q6W5P4 2/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8776704 0.84 RAB9A (0.45) LDHATSHRCA1CA2L3MBTL1
SCHEMBL28898941 0.84 RAB9A (0.45) LDHATSHRCA1CA2L3MBTL1
SCHEMBL8776664 0.84 RAB9A (0.45) LDHATSHRCA1CA2L3MBTL1
SCHEMBL6478492 0.81 LDHA (0.50) LDHAAKR1C3AKR1C2PTGS2PTGS1
SCHEMBL7082950 0.81 LDHA (0.50) LDHAAKR1C3AKR1C2PTGS2PTGS1
SCHEMBL23298286 0.81 LDHA (0.50) LDHAAKR1C3AKR1C2PTGS2PTGS1
SCHEMBL30404277 0.81 LDHA (0.50) LDHAAKR1C3AKR1C2PTGS2PTGS1
SCHEMBL8776709 0.80 ALOX15 (0.49) TSHRL3MBTL1ALDH1A1NPSR1NPC1
SCHEMBL8776680 0.80 ALOX15 (0.49) TSHRL3MBTL1ALDH1A1NPSR1NPC1
SCHEMBL18325177 0.80 AKR1C3 (0.51) LDHAAKR1C3AKR1C2PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0447938-B1 Process for preparing 2-halogeno-3-hydroxy-3-phenyl-propionic acid ester compounds TANABE SEIYAKU CO (JP) 1995-10-18 EP claimed
US-5204248-A Enzymatic reduction of corresponding oxo derivative; intermediate for diltiazem TANABE SEIYAKU CO., LTD. (JP) 1993-04-20 US claimed
EP-0447938-A1 Process for preparing 2-halogeno-3-hydroxy-3-phenyl-propionic acid ester compounds TANABE SEIYAKU CO., LTD. (JP) 1991-09-25 EP claimed
CN-113789353-A Preparation method of (2S,3S) -2-chloro-3-hydroxy ester compound 复旦大学 2021-12-14 CN disclosed
US-5081240-A PROCESS FOR THE PREPARATION OF BENZOTHIAZEPIN-ONE DERIVATIVES SANOFI (FR) 1992-01-14 US disclosed