SCHEMBL9186325

SCHEMBL9186325

CC(C)(C)OC(=O)N(CCCNc1ccccc1)CCCNc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA14 Q9ULX7 1/20 0.55
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
HDAC3 O15379 2/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC2 Q92769 2/20 0.44
NCOR2 Q9Y618 2/20 0.44
CCR6 P51684 1/20 0.42
PAX8 Q06710 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
METAP2 P50579 1/20 0.40
SSTR4 P31391 1/20 0.39
BACE1 P56817 1/20 0.37
CKS1B P61024 1/20 0.37
SKP1 P63208 1/20 0.37
SKP2 Q13309 1/20 0.37
REN P00797 1/20 0.37
TRPV4 Q9HBA0 1/20 0.37
AKT1 P31749 2/20 0.36
CACNA1B Q00975 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9189125 0.97 CA14 (0.56) CA14ALDH1A1MAPTHDAC3HDAC1
SCHEMBL12311224 0.81 GBA1 (0.44) ALDH1A1MAPTHDAC3HDAC1HDAC2
SCHEMBL9188875 0.81 CCR6 (0.66) CA14HDAC3HDAC1HDAC2NCOR2
SCHEMBL30941664 0.80 ROCK2 (0.41) CA14HDAC3HDAC1HDAC2NCOR2
SCHEMBL9180351 0.79 CA14 (0.50) CA14ALDH1A1MAPTSSTR4
SCHEMBL9891452 0.78 ALDH1A1 (0.48) ALDH1A1MAPTHDAC3HDAC1HDAC2
SCHEMBL7983925 0.77 L3MBTL1 (0.46) CA14HDAC3HDAC1HDAC2NCOR2
SCHEMBL1844315 0.77 L3MBTL1 (0.46) CA14HDAC3HDAC1HDAC2NCOR2
SCHEMBL10126784 0.77 MEN1 (0.53) ALDH1A1MAPTMETAP2
SCHEMBL25046666 0.76 L3MBTL1 (0.45) CA14HDAC3HDAC1HDAC2NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497202-B1 Polyamine thiols as radioprotective agents MERRELL DOW PHARMA (US) 1995-09-13 EP disclosed
US-5217964-A POLYAMINE THIOLS AS RADIOPROTECTIVE AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-08 US disclosed
EP-0497202-A1 Polyamine thiols as radioprotective agents MERRELL DOW PHARMACEUTICALS INC. (US) 1992-08-05 EP disclosed