SCHEMBL9188680

SCHEMBL9188680

CS(=O)(=O)OCCN(N(S(C)(=O)=O)S(C)(=O)=O)S(=O)(=O)c1ccc(Br)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.37
PLCG1 P19174 1/20 0.35
GAA P10253 1/20 0.33
ALDH1A1 P00352 3/20 0.33
LMNA P02545 3/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CA2 P00918 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
TP53 P04637 2/20 0.32
THRB P10828 2/20 0.32
KDM4E B2RXH2 2/20 0.32
GPR55 Q9Y2T6 1/20 0.32
USP2 O75604 1/20 0.32
MMP9 P14780 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9186665 0.87 CNR2 (0.40) ALDH1A1LMNAMAPTKEAP1NFE2L2
SCHEMBL9185920 0.86 CA12 (0.41) ALDH1A1MEN1KMT2ACA2ALOX15
SCHEMBL9188254 0.85 TDP1 (0.41) ALDH1A1LMNAKMT2A
SCHEMBL9285790 0.84 APLNR (0.44) ALDH1A1LMNAKEAP1NFE2L2
SCHEMBL9187495 0.81 SIGMAR1 (0.43) SIGMAR1PLCG1ALDH1A1MEN1KMT2A
SCHEMBL9190309 0.74 USP2 (0.46) ALDH1A1LMNAKDM4EUSP2MMP9
SCHEMBL18992740 0.72 ALDH1A1 (0.38) SIGMAR1PLCG1GAAALDH1A1LMNA
SCHEMBL22804712 0.71 TSHR (0.38) SIGMAR1PLCG1ALDH1A1LMNAMAPT
SCHEMBL5441671 0.68 CNR2 (0.50) ALDH1A1LMNAMAPTSMN1; SMN2
SCHEMBL9188734 0.67 CA12 (0.46) ALDH1A1LMNAMEN1KMT2ACA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0416286-B1 Sulfonylhydrazines and their use as antineoplastic agents and as antitrypanosomal agents UNIV YALE (US) 1995-08-09 EP disclosed
US-5214068-A Anticarcinogenic agents YALE UNIVERSITY (US) 1993-05-25 US disclosed
US-5101072-A Anticancer agents, trypanocides YALE UNIVERSITY (US) 1992-03-31 US disclosed
EP-0416286-A1 Sulfonylhydrazines and their use as antineoplastic agents and as antitrypanosomal agents YALE UNIVERSITY (US) 1991-03-13 EP disclosed