SCHEMBL9192052

SCHEMBL9192052

C=CCCc1c(C(=O)O)cccc1-c1ccc(C#N)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 8/20 0.37
CYP11B1 P15538 7/20 0.37
SLC22A12 Q96S37 1/20 0.37
ACMSD Q8TDX5 1/20 0.36
XDH P47989 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
STAT3 P40763 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35
TUBB3 Q13509 1/20 0.35
TUBB2A Q13885 1/20 0.35
TUBB8 Q3ZCM7 1/20 0.35
TUBA3E Q6PEY2 1/20 0.35
TUBA1A Q71U36 1/20 0.35
TUBA1C Q9BQE3 1/20 0.35
TUBB6 Q9BUF5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8676486 0.85 SYK (0.45) CYP11B2CYP11B1SLC22A12XDHCD274
SCHEMBL8678083 0.83 LTB4R2 (0.43) CYP11B2CYP11B1SLC22A12CD274
SCHEMBL8678897 0.83 SYK (0.43) CYP11B2CYP11B1SLC22A12ACMSDCD274
SCHEMBL8678448 0.83 RARB (0.47) CYP11B2CYP11B1SLC22A12CD274
SCHEMBL9192050 0.83 CYP11B2 (0.37) CYP11B2CYP11B1SLC22A12
SCHEMBL9192514 0.81 SLC22A12 (0.40) CYP11B2CYP11B1SLC22A12
SCHEMBL9186976 0.77 MCL1 (0.44) CYP11B2CYP11B1
SCHEMBL9193119 0.76 XDH (0.43) CYP11B2CYP11B1SLC22A12XDH
SCHEMBL28844938 0.72 ALDH1A1 (0.43)
SCHEMBL4650767 0.71 RARB (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0464648-B1 4-Cyano-3-fluorophenyl esters HOFFMANN LA ROCHE (CH) 1995-12-06 EP disclosed
EP-0464648-A1 4-Cyano-3-fluorophenyl esters F. HOFFMANN-LA ROCHE AG (CH) 1992-01-08 EP disclosed